EP 1169306 A1 20020109 - DIBENZOAZULENE DERIVATIVES FOR TREATING THROMBOSIS, OSTEOPOROSIS, ARTERIOSCLEROSIS
Title (en)
DIBENZOAZULENE DERIVATIVES FOR TREATING THROMBOSIS, OSTEOPOROSIS, ARTERIOSCLEROSIS
Title (de)
DIBENZOAZULENDERIVATE ZUR BEHANDLUNG VON THROMBOSE, OSTEOPOROSE, ARTERIOSKLEROSE
Title (fr)
DERIVES DE DIBENZOAZULENE POUR LE TRAITEMENT DE LA THROMBOSE, DE L'OSTEOPOROSE ET DE L'ARTERIOSCLEROSE
Publication
Application
Priority
- DE 19916837 A 19990414
- EP 0002925 W 20000401
Abstract (en)
[origin: US6521646B1] Compounds of the formula (I) and their physiologically acceptable salts and solvates are useful as integrin-inhibiting substances. They are especially useful in the prophylaxis and treatment of cardiovascular disorders, of thrombosis, cardiac infarction, coronary heart diseases, arteriosclerosis, osteoporosis, in pathological conditions that are caused or propagated by angiogenesis and in tumor therapy.
IPC 1-7
IPC 8 full level
C07D 239/14 (2006.01); A61K 31/4402 (2006.01); A61K 31/505 (2006.01); A61P 3/10 (2006.01); A61P 7/02 (2006.01); A61P 9/00 (2006.01); A61P 9/10 (2006.01); A61P 13/12 (2006.01); A61P 17/06 (2006.01); A61P 19/00 (2006.01); A61P 19/02 (2006.01); A61P 19/10 (2006.01); A61P 27/02 (2006.01); A61P 27/06 (2006.01); A61P 29/00 (2006.01); A61P 31/04 (2006.01); A61P 31/10 (2006.01); A61P 31/12 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07C 69/00 (2006.01); C07D 213/74 (2006.01)
CPC (source: EP KR US)
A61P 3/10 (2017.12 - EP); A61P 7/02 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 17/06 (2017.12 - EP); A61P 19/00 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 19/10 (2017.12 - EP); A61P 27/02 (2017.12 - EP); A61P 27/06 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 31/04 (2017.12 - EP); A61P 31/10 (2017.12 - EP); A61P 31/12 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07C 69/757 (2013.01 - EP KR US); C07D 213/74 (2013.01 - EP KR US); C07C 2603/40 (2017.04 - EP US)
Citation (search report)
See references of WO 0063178A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
US 6521646 B1 20030218; AR 023496 A1 20020904; AU 3817400 A 20001102; BR 0009690 A 20020108; CA 2367359 A1 20001026; CN 1345312 A 20020417; CZ 20013704 A3 20020213; DE 19916837 A1 20001019; EP 1169306 A1 20020109; HU P0200643 A2 20020729; HU P0200643 A3 20031028; JP 2002542231 A 20021210; KR 20010102570 A 20011115; MX PA01010294 A 20020506; NO 20014976 D0 20011012; NO 20014976 L 20011012; PL 350354 A1 20021202; RU 2001129708 A 20040227; SK 14342001 A3 20020404; WO 0063178 A1 20001026; ZA 200109343 B 20030430
DOCDB simple family (application)
US 95881201 A 20011015; AR P000101738 A 20000414; AU 3817400 A 20000401; BR 0009690 A 20000401; CA 2367359 A 20000401; CN 00805748 A 20000401; CZ 20013704 A 20000401; DE 19916837 A 19990414; EP 0002925 W 20000401; EP 00917037 A 20000401; HU P0200643 A 20000401; JP 2000612271 A 20000401; KR 20017011575 A 20010912; MX PA01010294 A 20000401; NO 20014976 A 20011012; PL 35035400 A 20000401; RU 2001129708 A 20000401; SK 14342001 A 20000401; ZA 200109343 A 20011113