Global Patent Index - EP 1171126 A4

EP 1171126 A4 20020327 - 6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE

Title (en)

6-AZAINDOLE COMPOUNDS AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE

Title (de)

6-AZAINDOLVERBINDUNGEN ALS ANTAGONISTEN DES GONADOTROPIN FREISETZENDES HORMONS

Title (fr)

COMPOSES 6-AZAINDOLE UTILISES COMME ANTAGONISTES D'UNE HORMONE LIBERANT LA GONADOTROPINE

Publication

EP 1171126 A4 20020327 (EN)

Application

EP 00917762 A 20000306

Priority

  • US 0005815 W 20000306
  • US 12364899 P 19990310

Abstract (en)

[origin: WO0053179A1] There are disclosed compounds of formula (I) and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men and women.

IPC 1-7

A61K 31/435; C07D 471/04

IPC 8 full level

C07D 471/04 (2006.01)

CPC (source: EP)

A61P 1/00 (2017.12); A61P 5/10 (2017.12); A61P 15/18 (2017.12); A61P 25/20 (2017.12); A61P 35/00 (2017.12); C07D 471/04 (2013.01)

Citation (search report)

  • [DX] US 5849764 A 19981215 - GOULET MARK [US], et al
  • [DX] US 5756507 A 19980526 - GOULET MARK [US], et al
  • [DX] US 5780437 A 19980714 - GOULET MARK [US], et al
  • [A] GOULET M T: "CHAPTER 18. GONADOTROPIN RELEASING HORMONE ANTAGONISTS", ANNUAL REPORTS IN MEDICINAL CHEMISTRY, SAN DIEGO, US, 1995, pages 169 - 177, XP002928176, ISSN: 0065-7743
  • See references of WO 0053179A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0053179 A1 20000914; AU 3868900 A 20000928; CA 2367116 A1 20000914; EP 1171126 A1 20020116; EP 1171126 A4 20020327; JP 2002538204 A 20021112

DOCDB simple family (application)

US 0005815 W 20000306; AU 3868900 A 20000306; CA 2367116 A 20000306; EP 00917762 A 20000306; JP 2000603668 A 20000306