EP 1171435 A2 20020116 - PYRIMIDINE-2-ONE DERIVATIVES AS INTEGRIN RECEPTOR LIGANDS

Title (en)

PYRIMIDINE-2-ONE DERIVATIVES AS INTEGRIN RECEPTOR LIGANDS

Title (de)

PYRIMIDIN-2-ON DERIVATE ALS INTEGRINREZEPTORLIGANDEN

Title (fr)

PYRIMIDINE-2-ONE DERIVES COMME LIGANDS DE RECEPTEURS D'INTEGRINE

Publication

EP 1171435 A2 20020116 (DE)

Application

EP 00920612 A 20000329

Priority

DE 19916719 A 19990413
DE 19962998 A 19991224
EP 0002746 W 20000329

Abstract (en)

[origin: WO0061551A2] The invention relates to novel compounds that bind to integrin receptor ligands. The invention also relates to the production thereof, to their use as integrin receptor ligands and to their use for treating diseases, to pharmaceutical preparations that contain said compounds and to pharmaceutical preparations that contain at least one additional active compound.

IPC 1-7

C07D 401/14; A61K 31/505; A61P 9/10; C07D 401/12; C07D 239/46; C07D 403/12; C07D 403/14; C07D 403/04; C07D 405/14; C07D 417/14; C07D 409/14; C07D 417/12

IPC 8 full level

C07D 239/36 (2006.01); A61K 31/505 (2006.01); A61K 45/00 (2006.01); A61K 45/06 (2006.01); A61P 3/14 (2006.01); A61P 7/02 (2006.01); A61P 9/10 (2006.01); A61P 9/12 (2006.01); A61P 13/12 (2006.01); A61P 17/02 (2006.01); A61P 17/06 (2006.01); A61P 19/08 (2006.01); A61P 19/10 (2006.01); A61P 29/00 (2006.01); A61P 31/04 (2006.01); A61P 31/12 (2006.01); A61P 33/00 (2006.01); A61P 35/00 (2006.01); C07D 239/34 (2006.01); C07D 239/60 (2006.01); C07D 401/04 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 403/12 (2006.01); C07D 403/14 (2006.01); C07D 405/04 (2006.01); C07D 405/14 (2006.01); C07D 409/14 (2006.01); C07D 417/12 (2006.01); C07D 417/14 (2006.01)

CPC (source: EP KR US)

A61K 45/06 (2013.01 - EP KR US); A61P 3/14 (2017.12 - EP); A61P 7/00 (2017.12 - EP); A61P 7/02 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 9/12 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 17/02 (2017.12 - EP); A61P 17/06 (2017.12 - EP); A61P 19/00 (2017.12 - EP); A61P 19/08 (2017.12 - EP); A61P 19/10 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 31/00 (2017.12 - EP); A61P 31/04 (2017.12 - EP); A61P 31/12 (2017.12 - EP); A61P 33/00 (2017.12 - EP); A61P 35/00 (2017.12 - EP); C07D 239/34 (2013.01 - EP KR US); C07D 401/04 (2013.01 - EP KR US); C07D 401/12 (2013.01 - EP KR US); C07D 401/14 (2013.01 - EP KR US); C07D 403/12 (2013.01 - EP KR US); C07D 403/14 (2013.01 - EP KR US); C07D 405/04 (2013.01 - EP KR US); C07D 405/14 (2013.01 - EP KR US); C07D 409/14 (2013.01 - EP KR US); C07D 417/12 (2013.01 - EP KR US); C07D 417/14 (2013.01 - EP US)

Citation (search report)

See references of WO 0061551A2

Citation (examination)

US 5849893 A 19981215 - LOEBBERDING ANTONIUS [DE], et al
EP 0761681 A2 19970312 - HOECHST AG [DE]
EP 0863150 A1 19980909 - BOEHRINGER MANNHEIM GMBH [DE]
WO 9640685 A1 19961219 - PERSEPTIVE BIOSYSTEMS INC [US]
ZECHEL ET AL., BIOORG.MED.CHEM.LETT., no. 12, 2002, pages 165 - 169
CHEMICAL ABSTRACTS, vol. 82, 1975, Columbus, Ohio, US; abstract no. 327
CHEMICAL ABSTRACTS, vol. 90, 1979, Columbus, Ohio, US; abstract no. 147604
DOEL ET AL., TETRAHEDRON, vol. 30, - 1974, pages 2755 - 2759

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0061551 A2 20001019; WO 0061551 A3 20001228; AU 4112900 A 20001114; BG 105979 A 20020628; BR 0009739 A 20020409; CA 2368049 A1 20001019; CN 1353706 A 20020612; CZ 20013678 A3 20020717; EP 1171435 A2 20020116; HK 1046279 A1 20030103; HU P0203338 A2 20030328; IL 145773 A0 20020725; JP 2002541243 A 20021203; JP 3936844 B2 20070627; KR 20010108499 A 20011207; MX PA01010232 A 20020327; NO 20014961 D0 20011012; NO 20014961 L 20011107; PL 351279 A1 20030407; SK 14102001 A3 20020702; TR 200102944 T2 20020821; US 7125883 B1 20061024

DOCDB simple family (application)

EP 0002746 W 20000329; AU 4112900 A 20000329; BG 10597901 A 20011004; BR 0009739 A 20000329; CA 2368049 A 20000329; CN 00807554 A 20000329; CZ 20013678 A 20000329; EP 00920612 A 20000329; HK 02107845 A 20021030; HU P0203338 A 20000329; IL 14577300 A 20000329; JP 2000610827 A 20000329; KR 20017013063 A 20011013; MX PA01010232 A 20000329; NO 20014961 A 20011012; PL 35127900 A 20000329; SK 14102001 A 20000329; TR 200102944 T 20000329; US 95849102 A 20020618