Global Patent Index - EP 1173184 A1

EP 1173184 A1 20020123 - para-BORONOPHENYLALANINE COMPLEXES WITH FRUCTOSE AND RELATED CARBOHYDRATES AND POLYOLS

Title (en)

para-BORONOPHENYLALANINE COMPLEXES WITH FRUCTOSE AND RELATED CARBOHYDRATES AND POLYOLS

Title (de)

para-BORONOPHENYLALANINKOMPLEXE MIT FRUKTOSE UND AHNLICHEN KOHLENHYDRATEN UND POLYOLEN

Title (fr)

COMPLEXES DE para-BORONOPHENYLALANINE CONTENANT DE LA FRUCTOSE ET GLUCIDES ET POLYOLS CORRESPONDANTS

Publication

EP 1173184 A1 20020123 (EN)

Application

EP 00918342 A 20000324

Priority

  • US 0007833 W 20000324
  • US 28284799 A 19990331

Abstract (en)

[origin: WO0057887A1] The present invention is directed to salt-free and essentially salt-free p-boronophenylalanine-carbohydrate or p-boronophenylalanine-polyol complexes, as well as methods for making such compounds. In addition, the present invention provides methods for substantially solubilizing freeze-dried p-boronophenylalanine-carbohydrate and p-boronophenylalanine-polyol complexes. The present invention further provides compositions and methods for enhancing the solubility of boronophenylalanine.

IPC 1-7

A61K 31/70; C07H 1/00; C07F 5/02; C07F 9/02

IPC 8 full level

C07H 23/00 (2006.01); C07B 59/00 (2006.01); C07F 5/02 (2006.01); C07H 1/00 (2006.01)

CPC (source: EP US)

C07B 59/005 (2013.01 - EP US); C07F 5/025 (2013.01 - EP US); C07H 1/00 (2013.01 - EP US)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0057887 A1 20001005; AT E279201 T1 20041015; AU 3917000 A 20001016; CA 2368634 A1 20001005; CA 2368634 C 20070626; DE 60014881 D1 20041118; EP 1173184 A1 20020123; EP 1173184 A4 20030502; EP 1173184 B1 20041013; JP 2002540159 A 20021126; JP 4643017 B2 20110302; US 6169076 B1 20010102

DOCDB simple family (application)

US 0007833 W 20000324; AT 00918342 T 20000324; AU 3917000 A 20000324; CA 2368634 A 20000324; DE 60014881 T 20000324; EP 00918342 A 20000324; JP 2000607637 A 20000324; US 28284799 A 19990331