EP 1175211 A2 20020130 - ANTICONVULSANT DERIVATIVES USEFUL IN TREATING COCAINE DEPENDENCY
Title (en)
ANTICONVULSANT DERIVATIVES USEFUL IN TREATING COCAINE DEPENDENCY
Title (de)
ANTIKONVULSIVE DERIVATE ZUR BEHANDLUNG VON COCAINABHÄNGIGKEIT
Title (fr)
DERIVES ANTI-CONVULSION UTILES POUR LE TRAITEMENT DE LA COCAINOMANIE
Publication
Application
Priority
- US 0011722 W 20000428
- US 13187799 P 19990430
Abstract (en)
[origin: WO0066108A2] Anticonvulsant derivatives useful in treating cocaine dependency are disclosed.
[origin: WO0066108A2] Anticonvulsant derivatives of formula (I) useful in treating cocaine dependency are disclosed. Formula (I) wherein X is Ch2 or oxygen; R1 is hydrogen or C1-C4 alkyl; and R2, R3, R4 and R5 are independently hydrogen or C1 -C3 alkyl and, when X is CH2, R4 and R5 may be alkene groups joined to form a benzene ring and, when X is oxygen, R2 and R3 and/or R4 and R5 together may be a methylenedioxy group of formula (II), wherein R6 and R7 are the same or different and are hydrogen, C1 -C3 alkyl or R6 and R7 together with the carbon to which they are attached are joined to form a cyclopentyl or cyclohexyl ring.
IPC 1-7
IPC 8 full level
A61K 31/255 (2006.01); A61K 31/35 (2006.01); A61K 31/7048 (2006.01); A61P 25/30 (2006.01); C07H 11/00 (2006.01)
CPC (source: EP)
A61K 31/255 (2013.01); A61K 31/35 (2013.01); A61K 31/7048 (2013.01); A61P 25/30 (2017.12)
Citation (search report)
See references of WO 0066108A2
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0066108 A2 20001109; WO 0066108 A3 20010111; AU 4685300 A 20001117; CA 2372083 A1 20001109; EP 1175211 A2 20020130; JP 2002543123 A 20021217; MX PA01011014 A 20030630
DOCDB simple family (application)
US 0011722 W 20000428; AU 4685300 A 20000428; CA 2372083 A 20000428; EP 00928651 A 20000428; JP 2000614993 A 20000428; MX PA01011014 A 20000428