Global Patent Index - EP 1181301 A1

EP 1181301 A1 20020227 - OLIGONUCLEOTIDE SYNTHESIS WITH LEWIS ACIDS AS ACTIVATORS

Title (en)

OLIGONUCLEOTIDE SYNTHESIS WITH LEWIS ACIDS AS ACTIVATORS

Title (de)

OLIGONUKLEOTID-SYNTHESE MIT LEWIS-SÄURE ALS AKTIVATOREN

Title (fr)

SYNTHESE D'OLIGONUCLEOTIDES UTILISANT DES ACIDES DE LEWIS COMME ACTIVATEURS

Publication

EP 1181301 A1 20020227 (EN)

Application

EP 00926516 A 20000508

Priority

  • US 0012530 W 20000508
  • US 32505599 A 19990603

Abstract (en)

[origin: WO0075157A1] A process for synthesizing oligonucleotides by phosphoramidite chemistry wherein the improvement is the use of Lewis acids as activators for formation of the phosphorous-oxygen bond.

IPC 1-7

C07H 19/04; C07H 21/00

IPC 8 full level

C07H 21/04 (2006.01); C07H 19/10 (2006.01); C07H 19/20 (2006.01); C07H 21/00 (2006.01)

CPC (source: EP)

C07H 19/10 (2013.01); C07H 19/20 (2013.01); C07H 21/00 (2013.01)

Citation (search report)

See references of WO 0075157A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0075157 A1 20001214; CA 2376016 A1 20001214; EP 1181301 A1 20020227; JP 2003514766 A 20030422; MX PA01012444 A 20020730

DOCDB simple family (application)

US 0012530 W 20000508; CA 2376016 A 20000508; EP 00926516 A 20000508; JP 2001502438 A 20000508; MX PA01012444 A 20000508