Global Patent Index - EP 1183265 A4

EP 1183265 A4 20040714 - NOVEL FABH ENZYME, COMPOSITIONS CAPABLE OF BINDING TO SAID ENZYME AND METHODS OF USE THEREOF

Title (en)

NOVEL FABH ENZYME, COMPOSITIONS CAPABLE OF BINDING TO SAID ENZYME AND METHODS OF USE THEREOF

Title (de)

NEUES FABH-ENZYM, ZUSAMMENSETZUNGEN, DIE DIESES ENZYM BINDEN KÖNNEN, UND METHODEN SEINER VERWENDUNG

Title (fr)

NOUVEL ENZYME FABH, COMPOSITIONS CAPABLES DE SE LIER A CET ENZYME ET METHODES D'UTILISATION ASSOCIEES

Publication

EP 1183265 A4 20040714 (EN)

Application

EP 00939638 A 20000607

Priority

  • US 0015659 W 20000607
  • US 13812499 P 19990607

Abstract (en)

[origin: WO0075169A1] A novel <i>E. coli</i> FabH crystalline structure is identified. Also disclosed are methods of identifying inhibitors of these enzymes and/or active sites, and inhibitors identified by these methods.

IPC 1-7

C07K 14/245; C12N 9/10; G01N 33/50

IPC 8 full level

C12N 9/00 (2006.01); C12N 9/10 (2006.01); C12Q 1/25 (2006.01); G01N 33/15 (2006.01); G01N 33/50 (2006.01); G06F 17/30 (2006.01); G16B 15/30 (2019.01); C12R 1/19 (2006.01); G06F 19/00 (2006.01); G06F 19/16 (2011.01)

CPC (source: EP US)

C12N 9/1029 (2013.01 - EP); G16B 15/30 (2019.01 - EP US); G16B 15/00 (2019.01 - EP); Y02A 90/10 (2017.12 - EP)

Citation (search report)

  • [PX] QIU X ET AL: "CRYSTAL STRUCTURE OF BETA-KETOACYL-ACYL CARRIER PROTEIN SYNTHASE III A KEY CONDENSING ENZYME IN BACTERIAL FATTY ACID BIOSYNTHESIS", JOURNAL OF BIOLOGICAL CHEMISTRY, AMERICAN SOCIETY OF BIOLOGICAL CHEMISTS, BALTIMORE, MD, US, vol. 274, no. 51, 17 December 1999 (1999-12-17), pages 36465 - 36471, XP002941899, ISSN: 0021-9258
  • [PX] JANSON CHERYL A ET AL: "Crystallization of Escherichia coli beta-ketoacyl-ACP synthase III and the use of a dry flash-cooling technique for data collection", ACTA CRYSTALLOGRAPHICA SECTION D BIOLOGICAL CRYSTALLOGRAPHY, vol. 56, no. 6, June 2000 (2000-06-01), pages 747 - 748, XP009031050, ISSN: 0907-4449
  • [PX] DAVIES CHRISTOPHER ET AL: "The 1.8 ANG crystal structure and active-site architecture of beta-ketoacyl-acyl carrier protein synthase III (FabH) from Escherichia coli", STRUCTURE (LONDON), vol. 8, no. 2, February 2000 (2000-02-01), pages 185 - 195, XP002280548, ISSN: 0969-2126
  • [PX] KHANDEKAR SANJAY S ET AL: "Expression, purification, and crystallization of the Escherichia coli selenomethionyl beta-ketoacyl-acyl carrier protein synthase III", BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, vol. 270, no. 1, 2 April 2000 (2000-04-02), pages 100 - 107, XP002280549, ISSN: 0006-291X
  • See references of WO 0075169A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0075169 A1 20001214; EP 1183265 A1 20020306; EP 1183265 A4 20040714; JP 2003505014 A 20030212

DOCDB simple family (application)

US 0015659 W 20000607; EP 00939638 A 20000607; JP 2001502450 A 20000607