EP 1185511 A2 20020313 - INHIBITORS OF FACTOR XA
Title (en)
INHIBITORS OF FACTOR XA
Title (de)
FAKTOR XA INHIBITOREN
Title (fr)
INHIBITEURS DU FACTEUR Xa
Publication
Application
Priority
- US 0014193 W 20000524
- US 13583899 P 19990524
Abstract (en)
[origin: WO0071516A2] Novel compounds, their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful <i>in vitro</i> or <i>in vivo</i> for preventing or treating coagulation disorders.
[origin: WO0071516A2] Compounds, e.g. described in claim 5, formula (I) and formula (II), where A-B is (1), their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful <i>in vitro</i> or <i>in vivo</i> for preventing or treating coagulation disorders.
IPC 1-7
C07D 207/16; C07D 211/60; C07C 311/39; C07D 403/04; C07D 401/04; C07D 413/04; C07D 243/08; C07D 241/04; A61P 7/00; A61K 31/40
IPC 8 full level
A61K 31/155 (2006.01); A61K 31/18 (2006.01); A61K 31/275 (2006.01); A61K 31/401 (2006.01); A61K 31/402 (2006.01); A61K 31/451 (2006.01); A61P 7/02 (2006.01); A61P 9/00 (2006.01); A61P 9/04 (2006.01); A61P 9/10 (2006.01); C07C 311/46 (2006.01); C07D 207/16 (2006.01); C07D 211/60 (2006.01); C07D 241/04 (2006.01); C07D 243/08 (2006.01); C07D 401/04 (2006.01); C07D 403/04 (2006.01); C07D 413/04 (2006.01)
CPC (source: EP)
A61P 7/00 (2017.12); A61P 7/02 (2017.12); A61P 9/00 (2017.12); A61P 9/04 (2017.12); A61P 9/10 (2017.12); C07C 311/46 (2013.01); C07D 207/16 (2013.01); C07D 211/60 (2013.01); C07D 241/04 (2013.01); C07D 243/08 (2013.01); C07D 401/04 (2013.01); C07D 403/04 (2013.01); C07D 413/04 (2013.01)
Citation (search report)
See references of WO 0071515A2
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0071516 A2 20001130; WO 0071516 A3 20010118; WO 0071516 B1 20010301; AU 5283600 A 20001212; AU 5284000 A 20001212; CA 2371904 A1 20001130; CA 2374788 A1 20001130; EP 1185511 A2 20020313; EP 1185512 A2 20020313; JP 2003500390 A 20030107; JP 2003500391 A 20030107; WO 0071515 A2 20001130; WO 0071515 A3 20010125
DOCDB simple family (application)
US 0014209 W 20000524; AU 5283600 A 20000524; AU 5284000 A 20000524; CA 2371904 A 20000524; CA 2374788 A 20000524; EP 00937698 A 20000524; EP 00937704 A 20000524; JP 2000619772 A 20000524; JP 2000619773 A 20000524; US 0014193 W 20000524