Global Patent Index - EP 1185511 A2

EP 1185511 A2 20020313 - INHIBITORS OF FACTOR XA

Title (en)

INHIBITORS OF FACTOR XA

Title (de)

FAKTOR XA INHIBITOREN

Title (fr)

INHIBITEURS DU FACTEUR Xa

Publication

EP 1185511 A2 20020313 (EN)

Application

EP 00937698 A 20000524

Priority

  • US 0014193 W 20000524
  • US 13583899 P 19990524

Abstract (en)

[origin: WO0071516A2] Novel compounds, their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful <i>in vitro</i> or <i>in vivo</i> for preventing or treating coagulation disorders.

[origin: WO0071516A2] Compounds, e.g. described in claim 5, formula (I) and formula (II), where A-B is (1), their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful <i>in vitro</i> or <i>in vivo</i> for preventing or treating coagulation disorders.

IPC 1-7

C07D 207/16; C07D 211/60; C07C 311/39; C07D 403/04; C07D 401/04; C07D 413/04; C07D 243/08; C07D 241/04; A61P 7/00; A61K 31/40

IPC 8 full level

A61K 31/155 (2006.01); A61K 31/18 (2006.01); A61K 31/275 (2006.01); A61K 31/401 (2006.01); A61K 31/402 (2006.01); A61K 31/451 (2006.01); A61P 7/02 (2006.01); A61P 9/00 (2006.01); A61P 9/04 (2006.01); A61P 9/10 (2006.01); C07C 311/46 (2006.01); C07D 207/16 (2006.01); C07D 211/60 (2006.01); C07D 241/04 (2006.01); C07D 243/08 (2006.01); C07D 401/04 (2006.01); C07D 403/04 (2006.01); C07D 413/04 (2006.01)

CPC (source: EP)

A61P 7/00 (2017.12); A61P 7/02 (2017.12); A61P 9/00 (2017.12); A61P 9/04 (2017.12); A61P 9/10 (2017.12); C07C 311/46 (2013.01); C07D 207/16 (2013.01); C07D 211/60 (2013.01); C07D 241/04 (2013.01); C07D 243/08 (2013.01); C07D 401/04 (2013.01); C07D 403/04 (2013.01); C07D 413/04 (2013.01)

Citation (search report)

See references of WO 0071515A2

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

WO 0071516 A2 20001130; WO 0071516 A3 20010118; WO 0071516 B1 20010301; AU 5283600 A 20001212; AU 5284000 A 20001212; CA 2371904 A1 20001130; CA 2374788 A1 20001130; EP 1185511 A2 20020313; EP 1185512 A2 20020313; JP 2003500390 A 20030107; JP 2003500391 A 20030107; WO 0071515 A2 20001130; WO 0071515 A3 20010125

DOCDB simple family (application)

US 0014209 W 20000524; AU 5283600 A 20000524; AU 5284000 A 20000524; CA 2371904 A 20000524; CA 2374788 A 20000524; EP 00937698 A 20000524; EP 00937704 A 20000524; JP 2000619772 A 20000524; JP 2000619773 A 20000524; US 0014193 W 20000524