EP 1192144 A1 20020403 - RHODANINE DERIVATIVES AND THEIR USE IN INHIBITING AND IMAGING AMYLOIDS
Title (en)
RHODANINE DERIVATIVES AND THEIR USE IN INHIBITING AND IMAGING AMYLOIDS
Title (de)
RHODANINDERIVATE UND IHRE VERWENDUNG ZUR INHIBIERUNG UND BILDGEBUNG VON AMYLOIDEN
Title (fr)
DERIVES DE LA RHODANINE ET LEUR UTILISATION POUR L'INHIBITION ET LA MISE EN IMAGES D'AMYLOIDES
Publication
Application
Priority
- US 0015072 W 20000531
- US 13854599 P 19990610
Abstract (en)
[origin: WO0076988A1] The present invention provides a method of treating Alzheimer's disease using a compound of Formula (I). Also provided is a method of inhibiting the aggregation of amyloid proteins using a compound of Formula (I) and a method of imaging amyloid deposits using substituted rhodanine derivatives.
IPC 1-7
C07D 277/36; C07D 417/06; C07D 417/10; C07D 417/14; A61K 31/426; A61K 31/427; A61K 51/04; A61P 25/28
IPC 8 full level
A61K 31/426 (2006.01); A61K 31/427 (2006.01); A61K 31/454 (2006.01); A61K 31/4725 (2006.01); A61K 49/00 (2006.01); A61K 51/00 (2006.01); A61K 51/04 (2006.01); A61P 3/10 (2006.01); A61P 21/00 (2006.01); A61P 25/00 (2006.01); A61P 25/28 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 277/20 (2006.01); C07D 277/36 (2006.01); C07D 417/06 (2006.01); C07D 417/10 (2006.01); C07D 417/14 (2006.01)
CPC (source: EP)
A61K 51/0453 (2013.01); A61K 51/0455 (2013.01); A61K 51/0459 (2013.01); A61P 3/10 (2017.12); A61P 21/00 (2017.12); A61P 25/00 (2017.12); A61P 25/28 (2017.12); A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07D 277/20 (2013.01); C07D 417/06 (2013.01); C07D 417/10 (2013.01); C07D 417/14 (2013.01)
Citation (search report)
See references of WO 0076988A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0076988 A1 20001221; AU 5455400 A 20010102; BR 0011440 A 20020319; CA 2370316 A1 20001221; EP 1192144 A1 20020403; JP 2003502321 A 20030121; MX PA01009863 A 20020506; TR 200103561 T2 20020422
DOCDB simple family (application)
US 0015072 W 20000531; AU 5455400 A 20000531; BR 0011440 A 20000531; CA 2370316 A 20000531; EP 00939472 A 20000531; JP 2001503846 A 20000531; MX PA01009863 A 20000531; TR 200103561 T 20000531