EP 1206470 A2 20020522 - PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF ISOXAZOLECARBOXAMIDES AND ANALOGUES
Title (en)
PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF ISOXAZOLECARBOXAMIDES AND ANALOGUES
Title (de)
VERFAHREN UND ZWISCHENPRODUKTE ZUR HERSTELLUNG VON ISOXAZOLCARBOXAMIDEN UND ANALOGEN
Title (fr)
METHODES EFFICACES DE PREPARATION D'INHIBITEURS DE PROTEASE DE RHINOVIRUS, INTERMEDIAIRES CLES ET REACTEUR A MEMBRANE CONTINUE UTILE DANS LEUR PREPARATION
Publication
Application
Priority
- US 0023032 W 20000823
- US 15036599 P 19990824
Abstract (en)
[origin: WO0114576A2] Efficient synthetic routes for the preparation of rhinovirus protease inhibitors of formula (I), key intermediates useful in those synthetic routes, as well as a continuous membrane reactor useful for those synthetic routes. These compounds of formula (I), as well as pharmaceutical compositions that contain these compounds, are suitable for treating patients or hosts infected with one or more picornaviruses.
[origin: WO0114576A2] Efficient synthetic routes for the preparation of rhinovirus protease inhibitors of formula (I), particulary (I'), key intermediates useful in those synthetic routes, as well as a continuous membrane reactor useful for those synthetic routes. These compounds of formula (I), as well as pharmaceutical compositions that contain these compounds, are suitable for treating patients or hosts infected with one or more picornaviruses.
IPC 1-7
C07D 413/12; C07D 261/18; C07C 309/65; C07C 303/28; C07C 69/732; C07C 59/56; C07C 271/22; C07C 229/36; C07C 51/347; C12P 17/14; C12P 7/42; C12P 1/00
IPC 8 full level
A61K 31/422 (2006.01); A61P 31/14 (2006.01); B01J 19/24 (2006.01); C07C 69/732 (2006.01); C07C 229/34 (2006.01); C07C 271/22 (2006.01); C07C 303/28 (2006.01); C07D 207/26 (2006.01); C07D 261/18 (2006.01); C07D 413/12 (2006.01); C12M 1/12 (2006.01); C12P 17/14 (2006.01); C12P 7/42 (2006.01); C07C 309/65 (2006.01)
CPC (source: EP)
A61P 31/14 (2018.01); B01J 19/2435 (2013.01); B01J 19/2475 (2013.01); C07C 69/732 (2013.01); C07C 229/34 (2013.01); C07C 271/22 (2013.01); C07C 303/28 (2013.01); C07D 261/18 (2013.01); C07D 413/12 (2013.01); B01J 2219/00033 (2013.01); B01J 2219/00099 (2013.01); B01J 2219/00103 (2013.01); B01J 2219/00159 (2013.01); B01J 2219/00162 (2013.01); B01J 2219/00177 (2013.01); C07B 2200/07 (2013.01)
C-Set (source: EP)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0114576 A2 20010301; WO 0114576 A3 20010830; WO 0114576 A8 20020620; WO 0114576 B1 20010927; AU 6797000 A 20010319; AU 778062 B2 20041111; BR 0013323 A 20020402; CA 2376509 A1 20010301; CN 1157391 C 20040714; CN 1382139 A 20021127; CN 1524960 A 20040901; CZ 2002634 A3 20020911; EP 1206470 A2 20020522; HK 1051363 A1 20030801; HU P0203315 A2 20030228; HU P0203315 A3 20031229; IL 147862 A0 20020814; JP 2003511350 A 20030325; KR 20020030795 A 20020425; MX PA02001947 A 20021031; PL 357162 A1 20040726; ZA 200200506 B 20030625
DOCDB simple family (application)
US 0023032 W 20000823; AU 6797000 A 20000823; BR 0013323 A 20000823; CA 2376509 A 20000823; CN 00812011 A 20000823; CN 200410005445 A 20000823; CZ 2002634 A 20000823; EP 00955830 A 20000823; HK 03103445 A 20030515; HU P0203315 A 20000823; IL 14786200 A 20000823; JP 2001518887 A 20000823; KR 20027002323 A 20020222; MX PA02001947 A 20000823; PL 35716200 A 20000823; ZA 200200506 A 20020121