EP 1216033 A1 20020626 - VASOPRESSIN ANTAGONIST FORMULATION AND PROCESS
Title (en)
VASOPRESSIN ANTAGONIST FORMULATION AND PROCESS
Title (de)
VASOPRESSIN-ANTAGONIST FORMULIERUNG UND VERFAHREN
Title (fr)
FORMULATION D'ANTAGONISTE DE LA VASOPRESSINE ET PROCEDE DE FABRICATION
Publication
Application
Priority
- US 0026369 W 20000926
- US 40577299 A 19990927
Abstract (en)
[origin: WO0122945A1] This invention provides novel formulations for N-[4-(5H-pyrrolo[2,1-c][1,4]benzodiazepin-10(11H)ylcarbonyl)-3-chlorophenyl]-5-fluoro-2-methyl-benzamide, or a pharmaceutically acceptable salt thereof, and processes for making them, the formulations comprising from about 1 % to about 20 % of active ingredient, from about 1 % to about 18 % of a surfactant component, from about 50 % to about 80 % of a component of one or more polyethylene glycols, from about 1 % to about 20 % of a component of one or more sucrose fatty acid esters and/or polyvinylpyrrolidone and, optionnaly, one or more pharmaceutically acceptable preservatives or antioxidants.
IPC 1-7
IPC 8 full level
A61K 9/48 (2006.01); A61K 31/5517 (2006.01); A61K 47/10 (2006.01); A61K 47/26 (2006.01); A61K 47/28 (2006.01); A61K 47/32 (2006.01); A61K 47/34 (2006.01); A61P 7/10 (2006.01); A61P 43/00 (2006.01)
CPC (source: EP KR)
A61K 9/4858 (2013.01 - EP); A61K 9/4866 (2013.01 - EP); A61K 31/5513 (2013.01 - KR); A61K 31/5517 (2013.01 - EP); A61P 7/10 (2018.01 - EP); A61P 13/00 (2018.01 - EP); A61P 43/00 (2018.01 - EP)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0122945 A1 20010405; AR 025780 A1 20021211; AU 7615000 A 20010430; BR 0014351 A 20020611; CA 2388474 A1 20010405; CN 1391466 A 20030115; CZ 20021083 A3 20020612; EA 200200414 A1 20021226; EP 1216033 A1 20020626; HK 1045109 A1 20021115; HU P0202972 A2 20021228; HU P0202972 A3 20030728; IL 148541 A0 20020912; JP 2003510269 A 20030318; KR 20020039354 A 20020525; MX PA02003189 A 20020930; NO 20021475 D0 20020325; NO 20021475 L 20020416; PL 354282 A1 20031229; ZA 200203312 B 20031231
DOCDB simple family (application)
US 0026369 W 20000926; AR P000105036 A 20000926; AU 7615000 A 20000926; BR 0014351 A 20000926; CA 2388474 A 20000926; CN 00816008 A 20000926; CZ 20021083 A 20000926; EA 200200414 A 20000926; EP 00965430 A 20000926; HK 02106544 A 20020905; HU P0202972 A 20000926; IL 14854100 A 20000926; JP 2001526157 A 20000926; KR 20027003931 A 20020326; MX PA02003189 A 20000926; NO 20021475 A 20020325; PL 35428200 A 20000926; ZA 200203312 A 20020425