Global Patent Index - EP 1235801 A2

EP 1235801 A2 2002-09-04 - SOLID PHARMACEUTICAL PREPARATION

Title (en)

SOLID PHARMACEUTICAL PREPARATION

Title (de)

FESTE ARZNEIZUBEREITUNG

Title (fr)

PREPARATION PHARMACEUTIQUE SOLIDE

Publication

EP 1235801 A2 (EN)

Application

EP 00977904 A

Priority

  • JP 0008283 W
  • JP 33954799 A
  • US 66157700 A

Abstract (en)

[origin: WO0140182A2] The present invention provides a solid preparation comprising a crystal of [3-[(2R)-[[(2R)-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]-1H-indol-7-yloxy]acetic acid (Compound A), especially a crystal of Compound A having a particle size of not larger than 100 mu m at the cumulative weight distribution value of 50 %, and not larger than 200 mu m at the cumulative weight distribution value of 95 %, preferably a solid preparation having the excellent stability and the content uniformity of Compound A, which is prepared by preparing granules of the crystal of Compound A with fillers, disintegrants and binders, and then followed by mixing said granules with external excipients.

IPC 1-7 (main, further and additional classification)

C07D 209/16; A61K 31/404; A61P 3/04

IPC 8 full level (invention and additional information)

A61K 9/14 (2006.01); A61K 9/20 (2006.01); A61K 31/404 (2006.01); A61P 3/04 (2006.01); A61P 3/10 (2006.01); A61P 43/00 (2006.01); C07D 209/14 (2006.01); C07D 209/16 (2006.01)

CPC (invention and additional information)

C07D 209/16 (2013.01)

Citation (search report)

See references of WO 0140182A3

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

EPO simple patent family

WO 0140182 A2 20010607; WO 0140182 A3 20020627; AU 1550501 A 20010612; CA 2391646 A1 20010607; CN 1433403 A 20030730; CZ 20021833 A3 20030212; EP 1235801 A2 20020904; HU 0203865 A2 20030328; HU 0203865 A3 20040528; IL 149635 D0 20021110; JP 2003515587 A 20030507; MX PA02005326 A 20030212; NO 20022541 A 20020729; NO 20022541 D0 20020529; NZ 519086 A 20031128; PL 356468 A1 20040628; SK 7362002 A3 20030204

INPADOC legal status


2009-07-03 [REG HK WD] APPLICATIONS WITHDRAWN, DEEMED TO BE WITHDRAWN, OR REFUSED AFTER PUBLICATION IN HONG KONG

- Document: HK 1046140

2005-02-09 [18W] APPLICATION WITHDRAWN

- Effective date: 20041214

2002-09-04 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20020628

2002-09-04 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A2

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

2002-09-04 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO:

- Free text: AL;LT PAYMENT 20020627;LV PAYMENT 20020627;MK;RO PAYMENT 20020627;SI PAYMENT 20020627