EP 1237895 A2 20020911 - PHOSPHORYLATION OF TERMINAL PRIMARY ALCOHOL GROUPS
Title (en)
PHOSPHORYLATION OF TERMINAL PRIMARY ALCOHOL GROUPS
Title (de)
PHOSPHORYLIERUNG VON TERMINALEN PRIMÄREN ALKOHOL- GRUPPEN
Title (fr)
PROCESSUS CHIMIQUES ET INTERMEDIAIRES
Publication
Application
Priority
- GB 0004527 W 20001128
- GB 9928499 A 19991203
Abstract (en)
[origin: WO0140236A2] The invention relates to chemical processes and chemical intermediates which are useful in the selective formation of a primary mono-phosphoryl group (-OPO(OH2)) in a terminal 1,2-diol-propanoyl (HO-CH2CH(OH)-CO-) containing system, and to chemical processes and chemical intermediates (and processes for their manufacture) particularly useful for the manufacture of anti-Gram positive oxazolidinone bacterial agents containing such functionality, in particular for the preparation of 5(R)-Isoxazol-3-yloxymethyl-3-(4-(1-(2(S) -hychoxy-3-phosphoryl-propanoyl)-1,2,5,6-tetrahydropyridy-4-il)3,5-difluorophenyl)oxazolidin-2-one.
IPC 1-7
C07F 9/09; C07F 9/6558; C07D 413/14; C07D 413/12; C07F 9/6574
IPC 8 full level
C07D 413/12 (2006.01); C07D 413/14 (2006.01); C07F 9/09 (2006.01); C07F 9/6518 (2006.01); C07F 9/6558 (2006.01); C07F 9/6574 (2006.01)
CPC (source: EP KR)
C07D 413/12 (2013.01 - EP); C07D 413/14 (2013.01 - EP); C07F 9/09 (2013.01 - KR); C07F 9/091 (2013.01 - EP); C07F 9/65583 (2013.01 - EP); C07F 9/65742 (2013.01 - EP)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 0140236 A2 20010607; WO 0140236 A3 20020510; AR 026700 A1 20030226; AU 1715601 A 20010612; AU 762241 B2 20030619; BG 106728 A 20030228; BR 0016087 A 20020806; CA 2395052 A1 20010607; CN 1433421 A 20030730; CO 5271712 A1 20030430; CZ 20021912 A3 20020814; EE 200200282 A 20030616; EP 1237895 A2 20020911; GB 9928499 D0 20000202; HU P0204052 A2 20030328; IL 149641 A0 20021110; IS 6401 A 20020528; JP 2003515539 A 20030507; KR 20020058072 A 20020712; MX PA02005396 A 20021129; NO 20022605 D0 20020531; NO 20022605 L 20020626; PL 364762 A1 20041213; SK 7862002 A3 20030204; ZA 200203876 B 20030815
DOCDB simple family (application)
GB 0004527 W 20001128; AR P000106370 A 20001201; AU 1715601 A 20001128; BG 10672802 A 20020520; BR 0016087 A 20001128; CA 2395052 A 20001128; CN 00818735 A 20001128; CO 00090190 A 20001124; CZ 20021912 A 20001128; EE P200200282 A 20001128; EP 00979764 A 20001128; GB 9928499 A 19991203; HU P0204052 A 20001128; IL 14964100 A 20001128; IS 6401 A 20020528; JP 2001540991 A 20001128; KR 20027007072 A 20020601; MX PA02005396 A 20001128; NO 20022605 A 20020531; PL 36476200 A 20001128; SK 7862002 A 20001128; ZA 200203876 A 20020515