EP 1239852 A2 20020918 - BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS
Title (en)
BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS
Title (de)
BISSULFONAMID-DERIVATE ALS ENZYM INHIBITOREN
Title (fr)
INHIBITEURS D'ENZYMES
Publication
Application
Priority
- GB 0003944 W 20001013
- GB 9924522 A 19991015
Abstract (en)
[origin: WO0128537A2] Bissulfonamide derivatives of formula (I) are capable of inhibiting: a) the biosynthesis of aromatic amino acids via the shikimate pathway and b) the catabolism of quinic acid, wherein: Ar is an aryl or heteroaryl group; R1 and R2 are the same or different and each represent hydrogen or alkyl or R1 and R2 together form a C1-C3 alkylene group, -CO- or -CS-; and R3 and R4 are the same or different and each represent -alkyl-aryl, -alkyl-heteroaryl, -alkenyl-aryl, -alkenyl-heteroaryl, -alkynyl-aryl-alkynyl-heterorayl, aryl or heteroaryl.
IPC 1-7
IPC 8 full level
A01N 41/06 (2006.01); A61K 31/145 (2006.01); A61K 31/18 (2006.01); A61K 31/381 (2006.01); A61K 31/422 (2006.01); A61K 31/425 (2006.01); A61K 31/426 (2006.01); A61K 31/4436 (2006.01); A61K 31/517 (2006.01); A61L 2/18 (2006.01); A61P 31/04 (2006.01); A61P 31/10 (2006.01); A61P 33/06 (2006.01); A61P 43/00 (2006.01); C07C 311/13 (2006.01); C07C 311/21 (2006.01); C07C 311/29 (2006.01); C07C 311/46 (2006.01); C07C 317/14 (2006.01); C07D 239/74 (2006.01); C07D 333/34 (2006.01); C07D 409/04 (2006.01); C07D 413/04 (2006.01); C07D 417/04 (2006.01)
CPC (source: EP KR)
A61K 31/18 (2013.01 - EP KR); A61P 31/04 (2017.12 - EP); A61P 31/10 (2017.12 - EP); A61P 33/06 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07C 311/13 (2013.01 - EP); C07C 311/21 (2013.01 - EP); C07C 311/29 (2013.01 - EP); C07C 311/46 (2013.01 - EP); C07C 317/14 (2013.01 - EP); Y02A 50/30 (2017.12 - EP)
Citation (search report)
See references of WO 0128537A2
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
DOCDB simple family (publication)
WO 0128537 A2 20010426; WO 0128537 A3 20010614; AU 7805400 A 20010430; CA 2387593 A1 20010426; EP 1239852 A2 20020918; GB 9924522 D0 19991215; JP 2003512319 A 20030402; KR 20020057973 A 20020712; ZA 200202897 B 20030414
DOCDB simple family (application)
GB 0003944 W 20001013; AU 7805400 A 20001013; CA 2387593 A 20001013; EP 00968096 A 20001013; GB 9924522 A 19991015; JP 2001531367 A 20001013; KR 20027004720 A 20020412; ZA 200202897 A 20020412