Global Patent Index - EP 1240169 A1

EP 1240169 A1 2002-09-18 - PEPTIDE BETA-TURN MIMETIC COMPOUNDS AND PROCESSES FOR MAKING THEM

Title (en)

PEPTIDE BETA-TURN MIMETIC COMPOUNDS AND PROCESSES FOR MAKING THEM

Title (de)

BETA-TURN MIMETISCHE PEPTID VERBINDUNGEN UND VERFAHREN ZU DEREN HERSTELLUNG

Title (fr)

COMPOSES MIMETIQUES DU VIRAGE-BETA PEPTIDIQUE ET PROCEDES DE FABRICATION DE CES DERNIERS

Publication

EP 1240169 A1 (EN)

Application

EP 00986673 A

Priority

  • US 0034832 W
  • US 17282399 P

Abstract (en)

[origin: WO0146197A1] The subject invention involves compounds having structure (I), wherein: (a) R1 is hydrogen or alkyl; and R2 is selected from hydrogen, alkyl, aryl, heterocyclyl, carboxy and its esters and amides; or R1 and R2 are attached and are together alkylene or heteroalkylene; (b) R4 is selected from aryl, heteroaryl, and alpha , beta -unsaturated conjugated aryl or heteroaryl; and (c) R5 is selected from hydrogen, alkyl, aryl, and heterocyclyl; and an optical isomer, diesteriomer, or enantiomer thereof; a salt, hydrate, ester, amide or imide thereof. The subject invention also includes libraries of such compounds, and processes for making the subject compounds and libraries.

IPC 1-7 (main, further and additional classification)

C07D 487/04; C07D 487/16; C07K 5/06

IPC 8 full level (invention and additional information)

C07D 487/04 (2006.01); C07D 487/14 (2006.01); C07K 1/04 (2006.01); C07K 5/02 (2006.01)

CPC (invention and additional information)

C07D 487/04 (2013.01); C07D 487/14 (2013.01); C07K 1/047 (2013.01); C07K 5/0215 (2013.01)

Citation (search report)

See references of WO 0146197A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

EPO simple patent family

WO 0146197 A1 20010628; AU 2286401 A 20010703; BR 0016518 A 20020924; CA 2393759 A1 20010628; CN 1413214 A 20030423; CO 5251420 A1 20030228; CZ 20022110 A3 20021113; EP 1240169 A1 20020918; HU 0300100 A2 20030528; IL 149834 D0 20021110; JP 2003518124 A 20030603; MX PA02006330 A 20021213; NO 20022953 A 20020619; NO 20022953 D0 20020619; PE 09552001 A1 20011011; PL 355971 A1 20040531

INPADOC legal status


2004-08-04 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20040122

2003-10-29 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20030911

2002-09-18 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20020621

2002-09-18 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

2002-09-18 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO

- Free text: AL;LT;LV;MK;RO;SI