EP 1240169 A1 20020918 - PEPTIDE BETA-TURN MIMETIC COMPOUNDS AND PROCESSES FOR MAKING THEM
Title (en)
PEPTIDE BETA-TURN MIMETIC COMPOUNDS AND PROCESSES FOR MAKING THEM
Title (de)
BETA-TURN MIMETISCHE PEPTID VERBINDUNGEN UND VERFAHREN ZU DEREN HERSTELLUNG
Title (fr)
COMPOSES MIMETIQUES DU VIRAGE-BETA PEPTIDIQUE ET PROCEDES DE FABRICATION DE CES DERNIERS
Publication
Application
Priority
- US 0034832 W 20001220
- US 17282399 P 19991221
Abstract (en)
[origin: WO0146197A1] The subject invention involves compounds having structure (I), wherein: (a) R1 is hydrogen or alkyl; and R2 is selected from hydrogen, alkyl, aryl, heterocyclyl, carboxy and its esters and amides; or R1 and R2 are attached and are together alkylene or heteroalkylene; (b) R4 is selected from aryl, heteroaryl, and alpha , beta -unsaturated conjugated aryl or heteroaryl; and (c) R5 is selected from hydrogen, alkyl, aryl, and heterocyclyl; and an optical isomer, diesteriomer, or enantiomer thereof; a salt, hydrate, ester, amide or imide thereof. The subject invention also includes libraries of such compounds, and processes for making the subject compounds and libraries.
IPC 1-7
IPC 8 full level
C07D 487/04 (2006.01); C07D 487/14 (2006.01); C07K 1/04 (2006.01); C07K 5/02 (2006.01)
CPC (source: EP KR)
C07D 487/04 (2013.01 - EP KR); C07D 487/14 (2013.01 - EP KR); C07K 1/047 (2013.01 - EP KR); C07K 5/0215 (2013.01 - EP KR)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 0146197 A1 20010628; AU 2286401 A 20010703; BR 0016518 A 20020924; CA 2393759 A1 20010628; CN 1413214 A 20030423; CO 5251420 A1 20030228; CZ 20022110 A3 20021113; EP 1240169 A1 20020918; HU P0300100 A2 20030528; IL 149834 A0 20021110; JP 2003518124 A 20030603; KR 20020062352 A 20020725; MX PA02006330 A 20021213; NO 20022953 D0 20020619; NO 20022953 L 20020619; PE 20010955 A1 20011011; PL 355971 A1 20040531
DOCDB simple family (application)
US 0034832 W 20001220; AU 2286401 A 20001220; BR 0016518 A 20001220; CA 2393759 A 20001220; CN 00817604 A 20001220; CO 00097142 A 20001221; CZ 20022110 A 20001220; EP 00986673 A 20001220; HU P0300100 A 20001220; IL 14983400 A 20001220; JP 2001547107 A 20001220; KR 20027007839 A 20020619; MX PA02006330 A 20001220; NO 20022953 A 20020619; PE 0013662000 A 20001219; PL 35597100 A 20001220