EP 1246819 A1 20021009 - A METHOD FOR THE PREPARATION OF SUBSTITUTED BENZENE DERIVATIVES
Title (en)
A METHOD FOR THE PREPARATION OF SUBSTITUTED BENZENE DERIVATIVES
Title (de)
VERFAHREN ZUR HERSTELLUNG SUBSTITUIERTER BENZENDERIVATE
Title (fr)
PROCEDE DE PREPARATION DE DERIVES DE BENZENE SUBSTITUE
Publication
Application
Priority
- DK 0000737 W 20001228
- DK PA199901886 A 19991230
- DK PA199901885 A 19991230
- DK PA200000942 A 20000616
Abstract (en)
[origin: WO0149681A1] A method for the preparation of selectively substituted benzene derivatives by application of solid phase synthesis is disclosed. In particular, the invention provides a novel method for the preparation of substituted benzene derivatives containing two or three groups bound to the benzene ring via nitrogen-, oxygen-, sulphur-, selenium- or carbon-carbon bonds, by application of solid phase chemistry alone or in combination with post cleavage solution phase derivatisation.
IPC 1-7
IPC 8 full level
C07D 209/14 (2006.01); C07D 243/04 (2006.01); C07D 295/04 (2006.01); C07D 295/08 (2006.01); C07D 295/12 (2006.01); C07D 403/06 (2006.01); C07D 403/12 (2006.01); C07D 405/12 (2006.01); C07D 405/14 (2006.01); C07D 413/12 (2006.01); C07D 413/14 (2006.01); C07D 471/04 (2006.01)
CPC (source: EP)
C07D 209/14 (2013.01); C07D 405/12 (2013.01)
Citation (search report)
See references of WO 0149681A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 0149681 A1 20010712; AU 2351701 A 20010716; EP 1246819 A1 20021009; JP 2003519227 A 20030617
DOCDB simple family (application)
DK 0000737 W 20001228; AU 2351701 A 20001228; EP 00987203 A 20001228; JP 2001550221 A 20001228