EP 1251134 A4 20030129 - NOVEL CARBAPENEM DERIVATIVES OF QUATERNARY SALT TYPE
Title (en)
NOVEL CARBAPENEM DERIVATIVES OF QUATERNARY SALT TYPE
Title (de)
NEUE CARBAPENEM-DERIVATE ALS QUATERNÄRES SALZ
Title (fr)
NOUVEAUX DERIVES DE CARBAPENEM DE TYPE SEL QUATERNAIRE
Publication
Application
Priority
- JP 0100529 W 20010126
- JP 2000017418 A 20000126
Abstract (en)
[origin: EP1251134A1] An objective of the present invention is to provide carbapenem derivatives which have potent antibiotic activity against MRSA, PRSP, Influenzavirus, and beta -lactamase-producing bacteria and are stable against DHP-1. The compounds according to the present invention are compounds represented by formula (I) or pharmaceutically acceptable salts thereof: <CHEM> wherein R<1> represents H or methyl; R<2> and R<3> each independently represent H, halogen, lower alkyl or the like; R<4> represents optionally substituted lower alkylthio or the like; and R<5> represents optionally substituted lower alkyl or the like.
IPC 1-7
C07D 519/00; A61K 31/429; A61P 31/04; A61K 31/415; A61K 31/495; A61K 31/535; A61K 31/445; A61K 31/47
IPC 8 full level
A61P 31/04 (2006.01); C07D 477/14 (2006.01); C07D 519/00 (2006.01); C07D 519/06 (2006.01)
CPC (source: EP US)
A61P 31/04 (2017.12 - EP); C07D 477/14 (2013.01 - EP US)
Citation (search report)
- No further relevant documents disclosed
- See references of WO 0155155A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
EP 1251134 A1 20021023; EP 1251134 A4 20030129; AU 2883301 A 20010807; CA 2398478 A1 20010802; US 2003022881 A1 20030130; US 6825187 B2 20041130; WO 0155155 A1 20010802
DOCDB simple family (application)
EP 01946865 A 20010126; AU 2883301 A 20010126; CA 2398478 A 20010126; JP 0100529 W 20010126; US 18218002 A 20020725