Global Patent Index - EP 1278744 A1

EP 1278744 A1 20030129 - HETEROBICYCLIC SULFONAMIDES AND THEIR USE AS PLATELET ADP RECEPTOR INHIBITORS

Title (en)

HETEROBICYCLIC SULFONAMIDES AND THEIR USE AS PLATELET ADP RECEPTOR INHIBITORS

Title (de)

HETEROBICYCLISCHE SULFONAMIDE UND IHRE VERWENDUNG ALS BLUTPLÄTTCHEN ADP REZEPTOR INHIBITOREN

Title (fr)

SULFONAMIDES HETEROBICYCLIQUES ET UTILISATION DE CELLES-CI COMME INHIBITEURS DE RECEPTEUR ADP DES PLAQUETTES

Publication

EP 1278744 A1 20030129 (EN)

Application

EP 01938998 A 20010504

Priority

  • US 0114441 W 20010504
  • US 20207500 P 20000505
  • US 23045600 P 20000906

Abstract (en)

[origin: WO0185722A1] The invention relates to novel compounds of formula (I) containing benzofused heterocyclic sulfonamide derivatives which are effective platelet ADP receptor inhibitors. Such compounds including pharmaceutically acceptable salts are useful in various pharmaceutical compositions for the prevention and/or treatment of cardiovascular disease particularly those related to thrombosis.

IPC 1-7

C07D 409/14; C07D 409/12; C07D 413/12; C07D 413/14; C07D 417/12; C07D 417/14; C07D 495/04; C07D 498/04; C07D 513/04; A61K 31/4184; A61K 31/423; A61K 31/428; A61K 31/4745; A61K 31/517; A61P 7/02

IPC 8 full level

A61K 31/4184 (2006.01); A61K 31/423 (2006.01); A61K 31/428 (2006.01); A61K 31/4365 (2006.01); A61K 31/437 (2006.01); A61K 31/517 (2006.01); A61P 7/00 (2006.01); A61P 7/02 (2006.01); A61P 9/02 (2006.01); A61P 9/10 (2006.01); A61P 9/14 (2006.01); A61P 43/00 (2006.01); C07D 409/12 (2006.01); C07D 409/14 (2006.01); C07D 413/12 (2006.01); C07D 413/14 (2006.01); C07D 417/12 (2006.01); C07D 417/14 (2006.01); C07D 495/04 (2006.01); C07D 498/04 (2006.01); C07D 513/04 (2006.01)

CPC (source: EP)

A61P 7/00 (2017.12); A61P 7/02 (2017.12); A61P 9/02 (2017.12); A61P 9/10 (2017.12); A61P 9/14 (2017.12); A61P 43/00 (2017.12); C07D 409/12 (2013.01); C07D 409/14 (2013.01); C07D 413/12 (2013.01); C07D 413/14 (2013.01); C07D 417/12 (2013.01); C07D 417/14 (2013.01); C07D 495/04 (2013.01); C07D 513/04 (2013.01)

Citation (search report)

See references of WO 0185722A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

DOCDB simple family (publication)

WO 0185722 A1 20011115; AU 6456601 A 20011120; CA 2408156 A1 20011115; EP 1278744 A1 20030129; HK 1050008 A1 20030606; JP 2003532728 A 20031105

DOCDB simple family (application)

US 0114441 W 20010504; AU 6456601 A 20010504; CA 2408156 A 20010504; EP 01938998 A 20010504; HK 03102259 A 20030328; JP 2001582323 A 20010504