EP 1298124 B1 20070228 - Method For the Preparation of Citalopram
Title (en)
Method For the Preparation of Citalopram
Title (de)
Verfahren zur Herstellung von Citalopram
Title (fr)
Procédé de préparation du citalopram
Publication
Application
Priority
DK 9900581 W 19991025
Abstract (en)
[origin: EP1298124A1] A method for the preparation of citalopram comprising reaction of a compound of Formula IV <CHEM> wherein R is C1-6 alkyl, acyl, C1-6 alkylsulfonyl or arylsulfonyl, with 3-(N,N-dimethylamino)-propyl magnesium halide, to prepare citalopram.
IPC 8 full level
C07C 255/56 (2006.01); A61K 31/343 (2006.01); A61P 25/24 (2006.01); C07C 253/30 (2006.01); C07D 307/87 (2006.01); C07D 307/93 (2006.01)
CPC (source: EP KR US)
A61K 31/343 (2013.01 - KR); A61P 25/24 (2018.01 - EP); C07C 255/56 (2013.01 - KR); C07D 307/87 (2013.01 - EP KR US)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated extension state (EPC)
AL LT LV MK RO SI
DOCDB simple family (publication)
EP 1298124 A1 20030402; EP 1298124 B1 20070228; AR 024518 A1 20021016; AT E277032 T1 20041015; AT E355268 T1 20060315; CA 2291133 A1 20010425; CA 2291133 C 20030617; CY 1107635 T1 20130418; CZ 292894 B6 20031217; DE 19983836 C1 20031023; DE 69920526 D1 20041028; DE 69920526 T2 20060223; DE 69935355 D1 20070412; DE 69935355 T2 20071108; DK 1228056 T3 20050124; DK 1298124 T3 20070709; EA 002801 B1 20021031; EA 200100593 A1 20011022; ES 2282365 T3 20071016; HK 1043129 A1 20020906; HK 1043129 B 20041021; HR P20020344 A2 20040229; HR P20020344 B1 20101031; HU P0200169 A2 20020629; HU P0200169 A3 20021128; IL 143875 A0 20020421; IL 143875 A 20080320; IL 176943 A0 20061210; IS 2260 B 20070615; IS 5970 A 20010615; KR 100505820 B1 20050803; KR 20010092799 A 20011027; NO 20071311 L 20010824; NZ 512406 A 20040130; PL 201056 B1 20090331; PL 349440 A1 20020729; PT 1228056 E 20050228; PT 1298124 E 20070531; SI 1228056 T1 20050228; SI 1298124 T1 20070831; SK 287140 B6 20100107; TR 200401456 T1 20050421; UA 72238 C2 20050215; US 2002177722 A1 20021128; US 6566540 B2 20030520
DOCDB simple family (application)
EP 02028326 A 19991025; AR P990105703 A 19991110; AT 02028326 T 19991025; AT 99950511 T 19991025; CA 2291133 A 19991025; CY 071100690 T 20070521; CZ 20022925 A 20020829; DE 19983836 A 19991025; DE 69920526 T 19991025; DE 69935355 T 19991025; DK 02028326 T 19991025; DK 99950511 T 19991025; EA 200100593 A 19991025; ES 02028326 T 19991025; HK 02105036 A 20020705; HR P20020344 A 20020419; HU P0200169 A 19991025; IL 14387501 A 20010620; IL 14387599 A 19991025; IL 17694306 A 20060718; IS 5970 A 20010615; KR 20017008100 A 20010623; NO 20071311 A 20070309; NZ 51240699 A 19991025; PL 34944099 A 19991025; PT 02028326 T 19991025; PT 99950511 T 19991025; SI 9930703 T 19991025; SI 9930960 T 19991025; SK 500082009 A 19991025; TR 200401456 T 19991025; UA 2001075224 A 19991025; US 13881102 A 20020503