EP 1299362 A1 20030409 - SELECTIVE MELANIN CONCENTRATING HORMONE-1 (MCH1) RECEPTOR ANTAGONISTS AND USES THEREOF
Title (en)
SELECTIVE MELANIN CONCENTRATING HORMONE-1 (MCH1) RECEPTOR ANTAGONISTS AND USES THEREOF
Title (de)
SELEKTIVE REZEPTORANTAGONISTEN DES MELANINKONZENTRIERENDEN HORMONS-1 (MCH1) UND IHRE ANWENDUNG
Title (fr)
ANTAGONISTES SELECTIFS DES RECEPTEURS (MCH1) D'HORMONE-1 DE CONCENTRATION DE LA MELANINE ET UTILISATION DE CEUX-CI
Publication
Application
Priority
- US 0121286 W 20010705
- US 61021300 A 20000705
Abstract (en)
[origin: WO0206245A1] This invention is directed to compounds which are selective antagonists for melanin concentrating hormone-1 (MCH1) receptors. The invention provides a pharmaceutical composition comprising a therapeutically effective amount of the compound of the invention and a pharmaceutically acceptable carrier. This invention provides a pharmaceutical composition made by combining a therapeutically effective amount of the compound of this invention and a pharmaceutically acceptable carrier. This invention further provides a process for making a pharmaceutical composition comprising combining a therapeutically effective amount of the compound of the invention and a pharmaceutically acceptable carrier. This invention also provides a method of modifying feeding behavior of a subject which comprises administering to the subject an amount of a compound of the invention effective to decrease the consumption of food by the subject. This invention further provides a method of treating a feeding disorder in a subject which comprises administering to the subject an amount of a compound of the invention effective to decrease the consumption of food by the subject. In an embodiment of the invention, the feeding disorder is bulimia, bulimia nervosa or obesity.
IPC 1-7
C07D 401/12; C07D 491/10; C07D 211/58; C07D 413/14; C07D 401/14; C07C 233/79; C07D 417/06; C07D 295/06; C07D 471/04; C07D 211/52; C07D 471/10; C07D 249/18; C07D 239/22; C07D 491/04; A61K 31/505; A61K 31/165; A61K 31/4188; A61K 31/4192; A61K 31/427; A61P 3/04; A61P 25/22; A61P 25/24
IPC 8 full level
A61K 9/02 (2006.01); A61K 9/08 (2006.01); A61K 9/20 (2006.01); A61K 31/165 (2006.01); A61K 31/166 (2006.01); A61K 31/4184 (2006.01); A61K 31/4188 (2006.01); A61K 31/4192 (2006.01); A61K 31/427 (2006.01); A61K 31/437 (2006.01); A61K 31/438 (2006.01); A61K 31/4468 (2006.01); A61K 31/451 (2006.01); A61K 31/4725 (2006.01); A61K 31/495 (2006.01); A61K 31/505 (2006.01); A61K 31/513 (2006.01); A61K 31/519 (2006.01); A61P 3/04 (2006.01); A61P 5/00 (2006.01); A61P 9/00 (2006.01); A61P 9/04 (2006.01); A61P 9/12 (2006.01); A61P 15/00 (2006.01); A61P 25/00 (2006.01); A61P 25/08 (2006.01); A61P 25/20 (2006.01); A61P 25/22 (2006.01); A61P 25/24 (2006.01); A61P 43/00 (2006.01); C07C 233/79 (2006.01); C07D 211/52 (2006.01); C07D 211/58 (2006.01); C07D 239/36 (2006.01); C07D 249/18 (2006.01); C07D 295/06 (2006.01); C07D 295/073 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 405/14 (2006.01); C07D 413/14 (2006.01); C07D 417/06 (2006.01); C07D 471/04 (2006.01); C07D 471/10 (2006.01); C07D 491/107 (2006.01); C07D 493/10 (2006.01)
CPC (source: EP)
A61K 31/165 (2013.01); A61K 31/4188 (2013.01); A61K 31/4192 (2013.01); A61K 31/427 (2013.01); A61K 31/505 (2013.01); A61P 3/04 (2017.12); A61P 5/00 (2017.12); A61P 9/00 (2017.12); A61P 9/04 (2017.12); A61P 9/12 (2017.12); A61P 15/00 (2017.12); A61P 25/00 (2017.12); A61P 25/08 (2017.12); A61P 25/20 (2017.12); A61P 25/22 (2017.12); A61P 25/24 (2017.12); A61P 43/00 (2017.12); C07C 233/79 (2013.01); C07D 211/52 (2013.01); C07D 211/58 (2013.01); C07D 239/36 (2013.01); C07D 249/18 (2013.01); C07D 295/073 (2013.01); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 413/14 (2013.01); C07D 417/06 (2013.01); C07D 471/04 (2013.01); C07D 471/10 (2013.01); C07D 493/10 (2013.01); C07C 2601/14 (2017.04)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 0206245 A1 20020124; AU 7319201 A 20020130; AU 783403 B2 20051020; CA 2384041 A1 20020124; EP 1299362 A1 20030409; EP 1299362 A4 20041103; JP 2004504303 A 20040212
DOCDB simple family (application)
US 0121286 W 20010705; AU 7319201 A 20010705; CA 2384041 A 20010705; EP 01952440 A 20010705; JP 2002512149 A 20010705