EP 1303271 A4 20040901 - OPHTHALMIC FORMULATION OF A SELECTIVE CYCLOOXYGENASE-2 INHIBITORY DRUG
Title (en)
OPHTHALMIC FORMULATION OF A SELECTIVE CYCLOOXYGENASE-2 INHIBITORY DRUG
Title (de)
OPTHALMISCHE ZUSAMMENSETZUNG ENTHALTEND CYCLOOXYGENASE-2-INHIBITOREN
Title (fr)
PREPARATION OPHTALMIQUE D'UN MEDICAMENT INHIBITEUR SELECTIF DE CYCLOOXYGENASE-2.
Publication
Application
Priority
- US 0122061 W 20010712
- US 21810100 P 20000713
- US 27928501 P 20010328
- US 29483801 P 20010531
- US 29638801 P 20010606
Abstract (en)
[origin: WO0205815A1] There is provided a pharmaceutical composition suitable for topical administration to an eye which contains a selective COX-2 inhibitory drug or nanoparticles of a drug of low water solubility, in a concentration effective for treatment and/or prophylaxis of a disorder in the eye, and one or more ophthalmically acceptable excipients that reduce rate of removal from the eye such that the composition has an effective residence time of about 2 to about 24 hours. Also provided is a method of treating and/or preventing a disorder in an eye, the method comprising administering to the eye a composition of the invention.
IPC 1-7
A61K 31/415; A61K 31/44; A61K 31/74; A61K 31/00; A61K 9/00; A61K 31/42; A61P 27/02
IPC 8 full level
C07D 237/16 (2006.01); A61K 9/00 (2006.01); A61K 31/12 (2006.01); A61K 31/122 (2006.01); A61K 31/352 (2006.01); A61K 31/353 (2006.01); A61K 31/365 (2006.01); A61K 31/38 (2006.01); A61K 31/415 (2006.01); A61K 31/42 (2006.01); A61K 31/435 (2006.01); A61K 31/44 (2006.01); A61K 31/4418 (2006.01); A61K 31/444 (2006.01); A61K 31/465 (2006.01); A61K 31/47 (2006.01); A61K 31/50 (2006.01); A61K 31/635 (2006.01); A61K 31/74 (2006.01); A61K 45/00 (2006.01); A61K 45/06 (2006.01); A61K 47/10 (2006.01); A61K 47/14 (2006.01); A61K 47/26 (2006.01); A61K 47/30 (2006.01); A61K 47/32 (2006.01); A61K 47/34 (2006.01); A61K 47/36 (2006.01); A61K 47/38 (2006.01); A61K 47/40 (2006.01); A61P 3/10 (2006.01); A61P 27/02 (2006.01); A61P 27/06 (2006.01); A61P 27/12 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); C07D 213/22 (2006.01); C07D 231/12 (2006.01); C07D 261/08 (2006.01); C07D 307/58 (2006.01); C07D 311/58 (2006.01); A61K 9/14 (2006.01); A61K 9/51 (2006.01)
CPC (source: EP US)
A61K 9/0048 (2013.01 - EP US); A61K 9/5138 (2013.01 - EP US); A61K 9/5161 (2013.01 - EP US); A61K 31/12 (2013.01 - EP US); A61K 31/122 (2013.01 - EP US); A61K 31/352 (2013.01 - EP US); A61K 31/353 (2013.01 - EP US); A61K 31/365 (2013.01 - EP US); A61K 31/38 (2013.01 - EP US); A61K 31/415 (2013.01 - EP US); A61K 31/42 (2013.01 - EP US); A61K 31/435 (2013.01 - EP US); A61K 31/44 (2013.01 - EP US); A61K 31/4418 (2013.01 - EP US); A61K 31/444 (2013.01 - EP US); A61K 31/465 (2013.01 - EP US); A61K 31/47 (2013.01 - EP US); A61K 31/50 (2013.01 - EP US); A61K 31/635 (2013.01 - EP US); A61K 31/74 (2013.01 - EP US); A61K 45/06 (2013.01 - EP US); A61K 47/10 (2013.01 - EP US); A61K 47/14 (2013.01 - EP US); A61K 47/26 (2013.01 - EP US); A61K 47/32 (2013.01 - EP US); A61K 47/38 (2013.01 - EP US); A61P 3/10 (2017.12 - EP); A61P 27/02 (2017.12 - EP); A61P 27/06 (2017.12 - EP); A61P 27/12 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61K 9/145 (2013.01 - EP US)
Citation (search report)
- [Y] WO 9631509 A1 19961010 - GLAXO GROUP LTD [GB], et al
- [Y] MASFERRER J L ET AL: "CYCLOOXYGENASE-2 INHIBITORS: A NEW APPROACH TO THE THERAPY OF OCULAR INFLAMMATION", SURVEY OF OPHTHALMOLOGY, SURVEY OF OPHTHALMOLOGY INC, XX, vol. 41, no. SUPPL 2, February 1997 (1997-02-01), pages 35 - 40, XP001027727, ISSN: 0039-6257
- See references of WO 0205815A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 0205815 A1 20020124; AR 033382 A1 20031217; AU 7590801 A 20020130; CA 2414780 A1 20020124; EP 1303271 A1 20030423; EP 1303271 A4 20040901; JP 2004528267 A 20040916; MX PA03000407 A 20041203; PE 20020146 A1 20020331; US 2002035264 A1 20020321
DOCDB simple family (application)
US 0122061 W 20010712; AR P010103304 A 20010712; AU 7590801 A 20010712; CA 2414780 A 20010712; EP 01953462 A 20010712; JP 2002511747 A 20010712; MX PA03000407 A 20010712; PE 2001000686 A 20010711; US 90409801 A 20010712