EP 1303482 A2 20030423 - N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES
Title (en)
N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES
Title (de)
N-SUBSTITUIERTE-1-AMINO-1,1-DIALKYLCARBONSÄUREDERIVATE
Title (fr)
DERIVES D'ACIDE 1-AMINO-1,1-DIALKYLCARBOXYLIQUE SUBSTITUES EN N
Publication
Application
Priority
- DE 10036121 A 20000725
- EP 0107596 W 20010703
Abstract (en)
[origin: WO0208177A2] The novel compounds of formula (I), wherein R<1>, R<2>, R<2'>, R<2">, R<3>, R<4>, R<5>, R<5'>, R<5">, R<5'''>, R<''''>, X, Y, U, V and W have the meanings given in patent claim no. 1, are inhibitors of the coagulation factors Xa and VIIa and can be used for treating thromboses, myocardial infarction, arteriosclerosis, inflammations, apoplexy, angina pectoris, restenosis following angioplasty, intermittent claudication, tumours, tumour diseases and/or tumour metastases.
IPC 1-7
C07C 311/46; C07D 271/06; A61K 31/165; A61K 31/18; A61P 9/00; A61P 35/00
IPC 8 full level
A61K 31/18 (2006.01); A61K 31/277 (2006.01); A61K 31/4245 (2006.01); A61P 7/02 (2006.01); A61P 9/00 (2006.01); A61P 9/10 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 35/04 (2006.01); C07B 61/00 (2006.01); C07C 311/46 (2006.01); C07D 211/66 (2006.01); C07D 213/40 (2006.01); C07D 271/06 (2006.01); C07D 309/14 (2006.01); C07D 335/02 (2006.01); C07D 401/12 (2006.01); C07D 405/12 (2006.01); C07D 409/12 (2006.01); C07D 413/12 (2006.01)
CPC (source: EP KR US)
A61P 7/02 (2018.01 - EP); A61P 9/00 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 35/00 (2018.01 - EP); A61P 35/04 (2018.01 - EP); C07C 311/46 (2013.01 - EP US); C07D 211/66 (2013.01 - EP US); C07D 213/40 (2013.01 - EP US); C07D 271/06 (2013.01 - EP US); C07D 309/14 (2013.01 - EP US); C07D 335/02 (2013.01 - EP US); C07D 401/12 (2013.01 - EP US); C07D 405/12 (2013.01 - EP US); C07D 409/12 (2013.01 - EP US); C07D 413/12 (2013.01 - EP KR US); C07C 2601/08 (2017.05 - EP US); C07C 2601/14 (2017.05 - EP US)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 0208177 A2 20020131; WO 0208177 A3 20020725; WO 0208177 A8 20020418; AR 029980 A1 20030723; AU 9369701 A 20020205; BR 0112771 A 20030624; CA 2418173 A1 20030123; CN 1443160 A 20030917; CZ 2003338 A3 20030514; DE 10036121 A1 20020207; EP 1303482 A2 20030423; HU P0302948 A2 20031229; JP 2004504375 A 20040212; KR 20030022163 A 20030315; MX PA03000664 A 20030606; NO 20030375 D0 20030124; NO 20030375 L 20030124; PL 358585 A1 20040809; SK 1512003 A3 20030701; US 2003162814 A1 20030828; ZA 200301471 B 20040629
DOCDB simple family (application)
EP 0107596 W 20010703; AR P010103542 A 20010725; AU 9369701 A 20010703; BR 0112771 A 20010703; CA 2418173 A 20010703; CN 01813181 A 20010703; CZ 2003338 A 20010703; DE 10036121 A 20000725; EP 01974078 A 20010703; HU P0302948 A 20010703; JP 2002514086 A 20010703; KR 20027017764 A 20021227; MX PA03000664 A 20010703; NO 20030375 A 20030124; PL 35858501 A 20010703; SK 1512003 A 20010703; US 33363303 A 20030123; ZA 200301471 A 20030224