Global Patent Index - EP 1307461 A2

EP 1307461 A2 20030507 - SUBSTITUTED PYRROLE COMPOUNDS AND THEIR USE AS SPLA2 INHIBITORS

Title (en)

SUBSTITUTED PYRROLE COMPOUNDS AND THEIR USE AS SPLA2 INHIBITORS

Title (de)

SUBSTITUIERTE PYRROL-VERBINDUNGEN UND IHRE VERWENDUNG ALS SPLA2-HEMMER

Title (fr)

NOUVEAUX INHIBITEURS DU SPLA 2?

Publication

EP 1307461 A2 20030507 (EN)

Application

EP 01958850 A 20010720

Priority

  • US 0121106 W 20010720
  • US 22339800 P 20000804

Abstract (en)

[origin: WO0212249A2] A class of novel substituted pyrrole is disclosed together with the use of such compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of Inflammatory Diseases such as septic shock.

IPC 1-7

C07D 495/04; A61K 31/407; A61P 29/00

IPC 8 full level

A61K 31/407 (2006.01); A61P 1/04 (2006.01); A61P 1/18 (2006.01); A61P 11/00 (2006.01); A61P 11/06 (2006.01); A61P 11/08 (2006.01); A61P 19/02 (2006.01); A61P 19/06 (2006.01); A61P 27/16 (2006.01); A61P 29/00 (2006.01); A61P 31/04 (2006.01); A61P 37/08 (2006.01); A61P 43/00 (2006.01); C07D 495/04 (2006.01)

CPC (source: EP)

A61P 1/04 (2017.12); A61P 1/18 (2017.12); A61P 11/00 (2017.12); A61P 11/06 (2017.12); A61P 11/08 (2017.12); A61P 19/02 (2017.12); A61P 19/06 (2017.12); A61P 27/16 (2017.12); A61P 29/00 (2017.12); A61P 31/04 (2017.12); A61P 37/08 (2017.12); A61P 43/00 (2017.12); C07D 495/04 (2013.01)

Citation (search report)

See references of WO 0212249A2

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

DOCDB simple family (publication)

WO 0212249 A2 20020214; WO 0212249 A3 20020718; AU 8046101 A 20020218; EP 1307461 A2 20030507; JP 2004505982 A 20040226

DOCDB simple family (application)

US 0121106 W 20010720; AU 8046101 A 20010720; EP 01958850 A 20010720; JP 2002518224 A 20010720