EP 1309549 A1 20030514 - ACETAMIDE DERIVATIVES AND THE USE THEREOF AS INHIBITORS OF COAGULATION FACTORS XA AND VIIA
Title (en)
ACETAMIDE DERIVATIVES AND THE USE THEREOF AS INHIBITORS OF COAGULATION FACTORS XA AND VIIA
Title (de)
ACETAMIDDERIVATE UND IHRE VERWENDUNG ALS INHIBITOREN DES KOAGULATIONSFAKTORS XA UND VIIA
Title (fr)
DERIVES D'ACETAMIDE ET LEUR UTILISATION EN TANT QU'INHIBITEURS DU FACTEUR DE COAGULATION XA ET VIIA
Publication
Application
Priority
- DE 10037146 A 20000729
- EP 0107594 W 20010703
Abstract (en)
[origin: WO0210127A1] The invention relates to novel compounds of formula (I) wherein R, R<1> and R<2> have the designation cited in patent claim 1. Said compounds are inhibitors of the coagulation factors Xa and VIIa, and can be used to treat thromboses, myocardial infarction, arteriosclerosis, inflammation, apoplexy, angina pectoris, restenosis after angioplasty, intermittent claudication, tumours, tumour diseases and/or tumour metastases.
IPC 1-7
C07C 333/08; C07C 317/44; C07C 311/16; C07C 257/18; C07D 413/12; C07D 271/06; C07D 213/30; C07D 211/46; A61K 31/18
IPC 8 full level
A61K 31/165 (2006.01); A61K 31/18 (2006.01); A61K 31/27 (2006.01); A61K 31/41 (2006.01); A61K 31/4245 (2006.01); A61K 31/4402 (2006.01); A61K 31/445 (2006.01); A61P 7/02 (2006.01); A61P 9/08 (2006.01); C07D 211/46 (2006.01); A61P 9/10 (2006.01); A61P 29/00 (2006.01); A61P 35/00 (2006.01); A61P 35/04 (2006.01); A61P 43/00 (2006.01); C07C 257/18 (2006.01); C07C 311/16 (2006.01); C07C 317/44 (2006.01); C07C 327/26 (2006.01); C07C 327/28 (2006.01); C07D 213/30 (2006.01); C07D 257/04 (2006.01); C07D 271/06 (2006.01)
CPC (source: EP KR US)
A61P 7/02 (2018.01 - EP); A61P 9/08 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 35/00 (2018.01 - EP); A61P 35/04 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07C 257/18 (2013.01 - EP US); C07C 311/16 (2013.01 - EP US); C07C 317/44 (2013.01 - EP US); C07C 333/08 (2013.01 - KR); C07D 271/06 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 0210127 A1 20020207; AR 029999 A1 20030723; AU 8194101 A 20020213; BR 0112813 A 20030701; CA 2417427 A1 20030127; CN 1444561 A 20030924; CZ 2003465 A3 20030514; DE 10037146 A1 20020207; EP 1309549 A1 20030514; HU P0301502 A2 20030828; JP 2004505106 A 20040219; KR 20030029531 A 20030414; MX PA03000780 A 20030604; NO 20030431 D0 20030128; NO 20030431 L 20030128; PL 358756 A1 20040823; SK 1972003 A3 20030603; US 2003187037 A1 20031002; ZA 200301633 B 20040622
DOCDB simple family (application)
EP 0107594 W 20010703; AR P010103584 A 20010727; AU 8194101 A 20010703; BR 0112813 A 20010703; CA 2417427 A 20010703; CN 01813469 A 20010703; CZ 2003465 A 20010703; DE 10037146 A 20000729; EP 01960449 A 20010703; HU P0301502 A 20010703; JP 2002516259 A 20010703; KR 20027017990 A 20021230; MX PA03000780 A 20010703; NO 20030431 A 20030128; PL 35875601 A 20010703; SK 1972003 A 20010703; US 34319603 A 20030129; ZA 200301633 A 20030227