EP 1353695 A2 20031022 - COMBINATIONS OF NICOTINIC ACID AND DERIVATIVES THEREOF AND STEROL ABSORPTION INHIBITOR(S) FOR THE TREATMENT OF VASCULAR INDICATIONS
Title (en)
COMBINATIONS OF NICOTINIC ACID AND DERIVATIVES THEREOF AND STEROL ABSORPTION INHIBITOR(S) FOR THE TREATMENT OF VASCULAR INDICATIONS
Title (de)
KOMBINATIONEN VON EINEM HEMMER DER STEROL-ABSORPTION UND NICOTINSÄURE ZUR BEHANDLUNG VON KARDIOVASKULÄREN INDIKATIONEN
Title (fr)
COMBINAISONS D'ACIDE NICOTINIQUE ET DE DERIVES DE CE DERNIER, INHIBITEUR(S) D'ABSORPTION DE STEROLS POUR LE TRAITEMENT DE CONDITIONS VASCULAIRES
Publication
Application
Priority
- US 0202004 W 20020125
- US 26427501 P 20010126
- US 32384201 P 20010921
Abstract (en)
[origin: WO02058685A2] The present invention provides compositions, therapeutic combinations and methods including: (a) at least one of nicotinic acid or derivatives thereof; and (b) at least one substituted azetidinone or substituted b-lactam sterol absorption inhibitor which can be useful for treating vascular conditions, diabetes, obesity and lowering plasma levels of sterols.
IPC 1-7
IPC 8 full level
C07D 205/08 (2006.01); A61K 31/216 (2006.01); A61K 31/22 (2006.01); A61K 31/337 (2006.01); A61K 31/366 (2006.01); A61K 31/397 (2006.01); A61K 31/40 (2006.01); A61K 31/404 (2006.01); A61K 31/4418 (2006.01); A61K 31/455 (2006.01); A61K 31/4965 (2006.01); A61K 31/655 (2006.01); A61K 31/7052 (2006.01); A61K 31/706 (2006.01); A61K 31/74 (2006.01); A61K 45/00 (2006.01); A61K 45/06 (2006.01); A61P 3/04 (2006.01); A61P 3/06 (2006.01); A61P 3/10 (2006.01); A61P 9/00 (2006.01); A61P 43/00 (2006.01)
CPC (source: EP US)
A61K 31/337 (2013.01 - EP US); A61K 31/395 (2013.01 - EP US); A61K 31/397 (2013.01 - EP US); A61K 31/455 (2013.01 - EP US); A61K 31/655 (2013.01 - EP US); A61K 31/7052 (2013.01 - EP US); A61K 31/74 (2013.01 - EP US); A61K 45/06 (2013.01 - EP US); A61P 3/04 (2017.12 - EP); A61P 3/06 (2017.12 - EP); A61P 3/10 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP)
Citation (search report)
See references of WO 02058685A2
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 02058685 A2 20020801; WO 02058685 A3 20030501; AR 034204 A1 20040204; AU 2002240050 A1 20020806; CA 2434488 A1 20020801; EP 1353695 A2 20031022; EP 1671650 A1 20060621; JP 2004517916 A 20040617; MX PA03006727 A 20031024; TW 200840563 A 20081016; US 2002183305 A1 20021205; US 2004097482 A1 20040520
DOCDB simple family (application)
US 0202004 W 20020125; AR P020100268 A 20020125; AU 2002240050 A 20020125; CA 2434488 A 20020125; EP 02705933 A 20020125; EP 06005831 A 20020125; JP 2002559019 A 20020125; MX PA03006727 A 20020125; TW 97121244 A 20020125; US 5764602 A 20020125; US 63990003 A 20030813