Global Patent Index - EP 1363890 A2

EP 1363890 A2 20031126 - MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF

Title (en)

MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF

Title (de)

MELANOCORTIN-4-REZEPTOR BINDENDE VERBINDUNGEN UND VERFAHREN ZU DEREN ANWENDUNG

Title (fr)

COMPOSES DE LIAISON AU RECEPTEUR DE LA MELANOCORTINE-4 ET PROCEDES D'UTILISATION DE TELS COMPOSES

Publication

EP 1363890 A2 20031126 (EN)

Application

EP 02718920 A 20020207

Priority

  • US 0203566 W 20020207
  • US 77846801 A 20010207

Abstract (en)

[origin: WO02062766A2] MC4-R binding compounds of the formula: B-Z-E (I) wherein B is an anchor moiety, Z is a central moiety, and E is a MC4-R interacting moiety are discussed. Methods of using the compounds to treat MC4-R associated disorders, such as disorders associated with weight loss, are also discussed.

IPC 1-7

C07D 235/06; C07D 239/06; C07D 233/20; A61K 31/4184; A61K 31/4164; A61K 31/505

IPC 8 full level

C07D 235/06 (2006.01); A61K 31/4164 (2006.01); A61K 31/4184 (2006.01); A61K 31/505 (2006.01); A61K 47/48 (2006.01); A61P 3/00 (2006.01); C07C 257/18 (2006.01); C07D 233/20 (2006.01); C07D 233/26 (2006.01); C07D 235/18 (2006.01); C07D 239/06 (2006.01); C07D 295/088 (2006.01); C07D 409/04 (2006.01)

CPC (source: EP)

A61K 31/4164 (2013.01); A61K 31/4184 (2013.01); A61K 31/505 (2013.01); A61K 47/54 (2017.07); A61P 3/00 (2017.12); C07C 257/18 (2013.01); C07D 233/20 (2013.01); C07D 233/26 (2013.01); C07D 235/18 (2013.01); C07D 239/06 (2013.01); C07D 295/088 (2013.01); C07D 409/04 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

DOCDB simple family (publication)

WO 02062766 A2 20020815; WO 02062766 A3 20021003; EP 1363890 A2 20031126; EP 1363890 A4 20090610

DOCDB simple family (application)

US 0203566 W 20020207; EP 02718920 A 20020207