Global Patent Index - EP 1380582 A1

EP 1380582 A1 20040114 - FSH mimetics for the treatment of infertility

Title (en)

FSH mimetics for the treatment of infertility

Title (de)

FSH Mimetika zur Behandlung von Infertilität

Title (fr)

Analogues de l'hormone de stimulation des follicules por traiter l'infertilité

Publication

EP 1380582 A1 20040114 (EN)

Application

EP 03023514 A 19990805

Priority

  • EP 99939686 A 19990805
  • US 9571298 P 19980807

Abstract (en)

The present invention provides non-peptidic amino derivatives, their therapeutic use as well as pharmaceutical compositions that possess activity as Follicle Stimulating Hormone (FSH) agonists and are useful in the for treatment of infertility. In particular, the invention provides cyclic and acyclic alpha- and beta-aminocarboxamides, more particularly tetrahydroisoquinolinecarboxamides, piperidinecarboxamides, pyrrolidinecarboxamides, and 2-amino-3-carboxamidopyridine derivatives.

IPC 1-7

C07D 401/12; A61K 31/445; A61K 31/40; C07D 405/14; C07D 405/12; C07K 5/06; C07D 471/04; A61P 5/24

IPC 8 full level

A61P 5/24 (2006.01); C07D 405/14 (2006.01); C07K 5/065 (2006.01); C07K 5/078 (2006.01); A61K 38/00 (2006.01)

CPC (source: EP)

A61P 5/24 (2017.12); C07D 405/14 (2013.01); C07K 5/06078 (2013.01); C07K 5/06139 (2013.01); A61K 38/00 (2013.01)

Citation (search report)

[A] US 5071836 A 19911210 - KOLAR CENEK [DE], et al

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

DOCDB simple family (publication)

EP 1380582 A1 20040114; EP 1380582 B1 20060614; DK 1380582 T3 20061204

DOCDB simple family (application)

EP 03023514 A 19990805; DK 03023514 T 19990805