Global Patent Index - EP 1423119 A4

EP 1423119 A4 20050413 - HETEROBICYCLES FKBP-LIGANDS

Title (en)

HETEROBICYCLES FKBP-LIGANDS

Title (de)

HETEROBICYCLEN FKBP-LIGANDEN

Title (fr)

LIGANDS DE LIAISON AVEC LES PROTEINES DE FIXATION DE FK-506 HETEROBICYCLES

Publication

EP 1423119 A4 20050413 (EN)

Application

EP 02731761 A 20020510

Priority

  • US 0214966 W 20020510
  • US 28982801 P 20010510

Abstract (en)

[origin: WO02089806A1] Diazabicyclo[3.3.1]nonane derivatives that inhibit the peptidyl-prolyl isomerase enzyme activity associated with FK-506 binding proteins (FKBP) are described for treating neurological disorders. Also described are compounds useful for preparing such inhibitors.

IPC 1-7

A61K 31/4995; A61K 31/5365; C07C 57/58; C07C 59/68; C07C 233/65; C07C 235/46; C07D 471/08; C07D 471/18; C07D 498/18

IPC 8 full level

A61K 31/439 (2006.01); A61K 31/4995 (2006.01); A61K 31/5365 (2006.01); A61K 31/5377 (2006.01); A61P 9/10 (2006.01); A61P 17/14 (2006.01); A61P 21/02 (2006.01); A61P 25/00 (2006.01); A61P 25/16 (2006.01); A61P 25/28 (2006.01); A61P 27/02 (2006.01); A61P 27/16 (2006.01); A61P 43/00 (2006.01); C07C 57/58 (2006.01); C07C 59/64 (2006.01); C07D 451/14 (2006.01); C07D 471/08 (2006.01); C07D 471/18 (2006.01); C07D 498/18 (2006.01); C07D 519/00 (2006.01)

CPC (source: EP)

A61P 9/10 (2017.12); A61P 17/14 (2017.12); A61P 21/02 (2017.12); A61P 25/00 (2017.12); A61P 25/16 (2017.12); A61P 25/28 (2017.12); A61P 27/02 (2017.12); A61P 27/16 (2017.12); A61P 43/00 (2017.12); C07C 57/58 (2013.01); C07C 59/64 (2013.01); C07D 471/08 (2013.01)

Citation (search report)

  • [PX] WO 0142245 A1 20010614 - BRISTOL MYERS SQUIBB CO [US]
  • [PX] WO 0232901 A2 20020425 - PFIZER PROD INC [US], et al
  • [E] WO 02060894 A2 20020808 - BRISTOL MYERS SQUIBB CO [US], et al
  • [X] GUO, C. ET AL: "A concise synthesis of AG5473/5507 utilizing N-acyliminium ion chemistry", TETRAHEDRON LETTERS, 41(28), 5307-5311 CODEN: TELEAY; ISSN: 0040-4039, 2000, XP004222061
  • See references of WO 02089806A1

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

DOCDB simple family (publication)

WO 02089806 A1 20021114; BR 0210060 A 20040817; CA 2446795 A1 20021114; EP 1423119 A1 20040602; EP 1423119 A4 20050413; JP 2004532854 A 20041028; MX PA03010255 A 20050307

DOCDB simple family (application)

US 0214966 W 20020510; BR 0210060 A 20020510; CA 2446795 A 20020510; EP 02731761 A 20020510; JP 2002586941 A 20020510; MX PA03010255 A 20020510