EP 1435910 B9 20100203 - NOVEL CYCLOSPORIN ANALOG MICROEMULSION PRECONCENTRATES
Title (en)
NOVEL CYCLOSPORIN ANALOG MICROEMULSION PRECONCENTRATES
Title (de)
NEUE CYCLOSPORIN-ANALOGE MIKROEMULSIONSVORKONZENTRATE
Title (fr)
NOUVEAUX PRECONCENTRES EN MICROEMULSION D'ANALOGUES DE CYCLOSPORINE
Publication
Application
Priority
- CA 0201561 W 20021017
- US 34620101 P 20011019
- US 37059702 P 20020405
Abstract (en)
[origin: WO03032949A1] The present invention relates to formulations containing cyclosporin analogs that are structurally similar to cyclosporin A, in particular isomeric mixtures of cyclosporin analogs that are structurally similar to cyclosporin A. The formulations form stable microemulsion preconcentrates and may provide superior drug bioavailability and/or may reduce one or more adverse effects associated with the administration of cyclosporin. Also disclosed are methods for using and preparing the formulations.
IPC 8 full level
A61K 9/10 (2006.01); A61K 9/107 (2006.01); A61K 9/00 (2006.01); A61K 9/48 (2006.01); A61K 38/00 (2006.01); A61K 38/13 (2006.01); A61K 47/10 (2006.01); A61K 47/14 (2006.01); A61K 47/22 (2006.01); A61K 47/30 (2006.01); A61K 47/34 (2006.01); A61K 47/44 (2006.01); A61P 29/00 (2006.01); A61P 37/06 (2006.01)
CPC (source: EP KR US)
A61K 9/0095 (2013.01 - EP US); A61K 9/107 (2013.01 - KR); A61K 9/1075 (2013.01 - EP US); A61K 9/4858 (2013.01 - EP US); A61K 38/13 (2013.01 - EP KR US); A61K 47/10 (2013.01 - EP US); A61P 1/04 (2018.01 - EP); A61P 1/16 (2018.01 - EP); A61P 3/10 (2018.01 - EP); A61P 7/00 (2018.01 - EP); A61P 7/04 (2018.01 - EP); A61P 7/06 (2018.01 - EP); A61P 9/00 (2018.01 - EP); A61P 11/00 (2018.01 - EP); A61P 11/06 (2018.01 - EP); A61P 13/12 (2018.01 - EP); A61P 17/00 (2018.01 - EP); A61P 17/04 (2018.01 - EP); A61P 17/06 (2018.01 - EP); A61P 17/14 (2018.01 - EP); A61P 19/02 (2018.01 - EP); A61P 19/08 (2018.01 - EP); A61P 21/00 (2018.01 - EP); A61P 21/04 (2018.01 - EP); A61P 25/00 (2018.01 - EP); A61P 27/02 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 31/12 (2018.01 - EP); A61P 37/00 (2018.01 - EP); A61P 37/02 (2018.01 - EP); A61P 37/06 (2018.01 - EP); A61P 37/08 (2018.01 - EP); C07K 7/00 (2013.01 - KR); C07K 7/64 (2013.01 - KR); C07K 7/645 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR IE IT LI LU MC NL PT SE SK TR
Designated extension state (EPC)
AL LT LV MK RO SI
DOCDB simple family (publication)
WO 03032949 A1 20030424; AR 036852 A1 20041006; AT E437629 T1 20090815; AU 2002333098 B2 20060316; BR 0213661 A 20041026; CA 2461730 A1 20030424; CA 2461730 C 20120515; CN 1274294 C 20060913; CN 1571657 A 20050126; CO 5580835 A2 20051130; DE 60233150 D1 20090910; DK 1435910 T3 20091109; EP 1435910 A1 20040714; EP 1435910 B1 20090729; EP 1435910 B9 20100203; EP 2116228 A1 20091111; ES 2330625 T3 20091214; HK 1062525 A1 20041112; HR P20040354 A2 20050228; HR P20040354 B1 20121031; IL 160761 A0 20040831; IL 160761 A 20101130; IL 195892 A 20130930; JP 2005506990 A 20050310; JP 2009073850 A 20090409; JP 2012158609 A 20120823; KR 100978836 B1 20100830; KR 20050037418 A 20050421; MA 26221 A1 20040701; ME P89008 A 20111220; MX PA04003623 A 20041202; MY 145753 A 20120330; NO 20042028 L 20040514; NZ 531946 A 20050930; PL 206018 B1 20100630; PL 370560 A1 20050530; PT 1435910 E 20090907; RU 2004110936 A 20050527; RU 2317067 C2 20080220; TN SN04070 A1 20060601; US 2003171264 A1 20030911; US 2006217309 A1 20060928; US 2009054311 A1 20090226; US 2011136744 A1 20110609; US 2014249092 A1 20140904; US 7060672 B2 20060613; US 7429562 B2 20080930; US 7829533 B2 20101109; ZA 200402268 B 20050525
DOCDB simple family (application)
CA 0201561 W 20021017; AR P020103917 A 20021017; AT 02801263 T 20021017; AU 2002333098 A 20021017; BR 0213661 A 20021017; CA 2461730 A 20021017; CN 02820641 A 20021017; CO 04035664 A 20040419; DE 60233150 T 20021017; DK 02801263 T 20021017; EP 02801263 A 20021017; EP 09166128 A 20021017; ES 02801263 T 20021017; HK 04105426 A 20040722; HR P20040354 A 20040419; IL 16076102 A 20021017; IL 16076104 A 20040305; IL 19589208 A 20081211; JP 2003535753 A 20021017; JP 2008287205 A 20081107; JP 2012118377 A 20120524; KR 20047005700 A 20021017; MA 27599 A 20040326; ME P89008 A 20021017; MX PA04003623 A 20021017; MY PI20023883 A 20021017; NO 20042028 A 20040514; NZ 53194602 A 20021017; PL 37056002 A 20021017; PT 02801263 T 20021017; RU 2004110936 A 20021017; TN SN04070 A 20040416; US 19719908 A 20080822; US 201414201872 A 20140309; US 27441902 A 20021017; US 37553206 A 20060313; US 94190710 A 20101108; ZA 200402268 A 20040323