EP 1448532 A1 20040825 - 5-PHENYLPYRIMIDINES, AGENTS COMPRISING THE SAME, METHOD FOR PRODUCTION AND USE THEREOF

Title (en)

5-PHENYLPYRIMIDINES, AGENTS COMPRISING THE SAME, METHOD FOR PRODUCTION AND USE THEREOF

Title (de)

5-PHENYLPYRIMIDINE, VERFAHREN ZU IHRER HERSTELLUNG, SIE ENTHALTENDE MITTEL UND IHRE VERWENDUNG

Title (fr)

5-PHENYLPYRIMIDINES, PROCEDE POUR LES PRODUIRE, AGENTS LES CONTENANT ET LEUR UTILISATION

Publication

EP 1448532 A1 20040825 (DE)

Application

EP 02787691 A 20021115

Priority

DE 10156279 A 20011119
EP 0212807 W 20021115

Abstract (en)

[origin: WO03043993A1] 5-Phenylpyrimidines of formula (I), where the substituents and the indices have the following meanings: R<1>, R<2> = H, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkinyl or haloalkinyl, where R<1> and R<2> together with the nitrogen atom to which they are bonded may form a saturated or unsaturated ring, interrupted by an ether, thio, sulphoxy or sulphonyl group and which can be substituted by one to four groups R<a> and/or R, R<3> = H, halo, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy, R<4> = H, halo, cyano, hydroxy, mercapto, azido, alkyl, alkenyl, alkinyl, haloalkyl, alkoxy, alkenyloxy, alkinyloxy, haloalkoxy, alkylthio, alkenylthio, alkinylthio, haloalkylthio, -ON=CR<a>R, -CR<c>=NOR<a>, -NR<c>N=CR<a>R, -NR<a>R, -NR<c>NR<a>R, -NOR<a>, -NR<c>C (=NR<c'>) NR<a>R, -NR<c>C (=0) NR<a>R, -NR<a>C (=0) R<c>, -NR<a>C (=NOR<c>)R<c'>, -OC (=0) R<c>, -C (=NOR<c>) NR<a>R, -CR<c> (=NNR<a>R), -C (=0) NR<a>R or -C (=0) R<c>, where R<a>,R,R<c> are as defined in the description, X = halo, alkyl, alkoxy or haloalkyl and m = a whole number from 1 to 5. The invention further relates to methods for production of the above compounds, agents containing the same and use thereof for the treatment of noxious mycoses.

IPC 1-7

C07D 239/46; C07D 239/48; C07D 239/42; C07D 239/52; C07D 403/12; A01N 43/54

IPC 8 full level

A01N 43/54 (2006.01); C07D 239/42 (2006.01); C07D 239/46 (2006.01); C07D 239/47 (2006.01); C07D 239/48 (2006.01); C07D 239/52 (2006.01); C07D 401/06 (2006.01); C07D 401/14 (2006.01); C07D 403/12 (2006.01)

CPC (source: EP KR US)

C07D 239/42 (2013.01 - EP US); C07D 239/46 (2013.01 - KR); C07D 239/47 (2013.01 - EP KR US); C07D 239/48 (2013.01 - EP US); C07D 239/52 (2013.01 - EP US); C07D 403/12 (2013.01 - EP US)

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR IE IT LI LU MC NL PT SE SK TR

DOCDB simple family (publication)

WO 03043993 A1 20030530; AU 2002352015 A1 20030610; AU 2002352015 B2 20080731; BR 0214253 A 20041214; CA 2467683 A1 20030530; CA 2467683 C 20110927; CN 1312134 C 20070425; CN 1606547 A 20050413; EA 010628 B1 20081030; EA 200400597 A1 20041230; EP 1448532 A1 20040825; HU P0402385 A2 20050329; HU P0402385 A3 20051028; IL 161893 A0 20051120; JP 2005514363 A 20050519; JP 4450625 B2 20100414; KR 100950632 B1 20100401; KR 20040079901 A 20040916; MX PA04004583 A 20040813; NZ 533265 A 20060526; PL 371059 A1 20050613; UA 78255 C2 20070315; US 2006148764 A1 20060706; US 2007149551 A1 20070628; US 7449471 B2 20081111; US 7465735 B2 20081216; ZA 200404835 B 20050620

DOCDB simple family (application)

EP 0212807 W 20021115; AU 2002352015 A 20021115; BR 0214253 A 20021115; CA 2467683 A 20021115; CN 02825535 A 20021115; EA 200400597 A 20021115; EP 02787691 A 20021115; HU P0402385 A 20021115; IL 16189302 A 20021115; JP 2003545630 A 20021115; KR 20047007560 A 20021115; MX PA04004583 A 20021115; NZ 53326502 A 20021115; PL 37105902 A 20021115; UA 20040604823 A 20021115; US 49528004 A 20040511; US 67786207 A 20070222; ZA 200404835 A 20040618