EP 1472219 A1 20041103 - NOVEL BENZOTHIAZINE AND BENZOTHIADIAZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
Title (en)
NOVEL BENZOTHIAZINE AND BENZOTHIADIAZINE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
Title (de)
NEUE BENZOTHIAZIN- UND BENZOTHIADIAZINDERIVATE, VERFAHREN ZU DEREN HERSTELLUNG UND PHARMAZEUTISCHE ZUSAMMENSETZUNGEN, DIE DIESE ENTHALTEN
Title (fr)
NOUVEAUX DERIVES DE BENZOTHIAZINE ET BENZOTHIADIAZINE, LEUR PROCEDE DE PREPARATION ET LES COMPOSITIONS PHARMACEUTIQUES QUI LES CONTIENNENT
Publication
Application
Priority
- FR 0204483 W 20021220
- FR 0116620 A 20011221
Abstract (en)
[origin: WO03053978A1] The invention concerns a compound of formula (I), wherein: R1 represents an aryl or heteroaryl; R2 represents hydrogen, halogen or a hydroxy; X represents oxygen or sulphur; Y represents oxygen, sulphur or NR wherein R represents hydrogen or an alkyl; A represents CR4R5 or NR4; R3 represents hydrogen, alkyl or cycloalkyl; R4 represents hydrogen or alkyl; or A represents nitrogen and forms with adjacent -CHR3-the cycle (a) wherein m represents 1, 2, or 3, R3 represents hydrogen or halogen; their isomers and their addition salts. Said compounds are useful as medicines, as AMPA modulators.
IPC 1-7
IPC 8 full level
C07D 285/24 (2006.01); A61K 31/549 (2006.01); A61P 25/00 (2006.01); A61P 25/08 (2006.01); A61P 25/14 (2006.01); A61P 25/18 (2006.01); A61P 25/22 (2006.01); A61P 25/24 (2006.01); A61P 25/28 (2006.01); C07D 279/02 (2006.01); C07D 513/04 (2006.01)
CPC (source: EP KR US)
A61P 25/00 (2017.12 - EP); A61P 25/08 (2017.12 - EP); A61P 25/14 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 25/22 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 25/28 (2017.12 - EP); C07D 279/02 (2013.01 - EP KR US); C07D 513/04 (2013.01 - EP KR US)
Citation (search report)
See references of WO 03053978A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR IE IT LI LU MC NL PT SE SI SK TR
DOCDB simple family (publication)
WO 03053978 A1 20030703; AR 038260 A1 20050112; AU 2002364673 A1 20030709; AU 2002364673 B2 20071122; BR 0214926 A 20041130; CA 2471120 A1 20030703; CN 1289508 C 20061213; CN 1606559 A 20050413; EA 007492 B1 20061027; EA 200400757 A1 20041028; EP 1472219 A1 20041103; FR 2833955 A1 20030627; FR 2833955 B1 20040130; GE P20063757 B 20060227; HK 1071746 A1 20050729; HU P0402583 A2 20050329; HU P0402583 A3 20090128; JP 2005518385 A 20050623; KR 100586684 B1 20060608; KR 20040073479 A 20040819; MA 27088 A1 20041220; MX PA04005839 A 20040910; NO 20042708 L 20040628; NZ 533329 A 20061027; PL 370166 A1 20050516; UA 78742 C2 20070425; US 2005065146 A1 20050324; US 7262189 B2 20070828; ZA 200404295 B 20050601
DOCDB simple family (application)
FR 0204483 W 20021220; AR P020105011 A 20021219; AU 2002364673 A 20021220; BR 0214926 A 20021220; CA 2471120 A 20021220; CN 02825674 A 20021220; EA 200400757 A 20021220; EP 02805406 A 20021220; FR 0116620 A 20011221; GE AP2002005643 A 20021220; HK 05104491 A 20050530; HU P0402583 A 20021220; JP 2003554694 A 20021220; KR 20047009200 A 20021220; MA 27717 A 20040604; MX PA04005839 A 20021220; NO 20042708 A 20040628; NZ 53332902 A 20021220; PL 37016602 A 20021220; UA 20040706009 A 20021220; US 49916404 A 20040615; ZA 200404295 A 20040601