Global Patent Index - EP 1494674 A1

EP 1494674 A1 20050112 - CARBOXIMIDE DERIVATIVES AS USEFUL URO-SELECTIVE ALPHA-1A ADRENOCEPTOR BLOCKERS

Title (en)

CARBOXIMIDE DERIVATIVES AS USEFUL URO-SELECTIVE ALPHA-1A ADRENOCEPTOR BLOCKERS

Title (de)

CARBOXIMID-DERIVATE ALS NÜTZLICHE UROSELEKTIVE ALPHA-1A ADRENOZEPTOR-BLOCKER

Title (fr)

DERIVES DE CARBOXIMIDE UTILES COMME BLOQUEURS UROSELECTIFS DU RECEPTEUR ADRENERGIQUE ALPHA-SB-1A

Publication

EP 1494674 A1 20050112 (EN)

Application

EP 02720343 A 20020408

Priority

IB 0201108 W 20020408

Abstract (en)

[origin: WO03084541A1] Novel carboximide derivatives, which selectively inhibit binding to the alpha >-1A< adrenergic receptor, a receptor which has been shown to be important in the treatment of benign prostatic hyperplasia. The compounds of the present invention are potentially useful in the treatment of benign prostatic hyperplasia.

IPC 1-7

A61K 31/495; C07D 295/13

IPC 8 full level

A61K 31/495 (2006.01); A61P 9/12 (2006.01); A61P 13/08 (2006.01); A61P 43/00 (2006.01); C07C 233/36 (2006.01); C07C 233/62 (2006.01); C07D 241/04 (2006.01); C07D 295/13 (2006.01)

CPC (source: EP)

A61P 9/12 (2017.12); A61P 13/08 (2017.12); A61P 43/00 (2017.12); C07D 295/13 (2013.01)

Designated contracting state (EPC)

AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

DOCDB simple family (publication)

WO 03084541 A1 20031016; AU 2002251409 A1 20031020; BR 0215686 A 20050222; CN 1627946 A 20050615; EA 200401335 A1 20060224; EP 1494674 A1 20050112; EP 1494674 A4 20060412; JP 2005532282 A 20051027; MX PA04009821 A 20041213

DOCDB simple family (application)

IB 0201108 W 20020408; AU 2002251409 A 20020408; BR 0215686 A 20020408; CN 02829097 A 20020408; EA 200401335 A 20020408; EP 02720343 A 20020408; JP 2003581781 A 20020408; MX PA04009821 A 20020408