EP 1494674 A4 20060412 - CARBOXIMIDE DERIVATIVES AS USEFUL URO-SELECTIVE ALPHA-1A ADRENOCEPTOR BLOCKERS
Title (en)
CARBOXIMIDE DERIVATIVES AS USEFUL URO-SELECTIVE ALPHA-1A ADRENOCEPTOR BLOCKERS
Title (de)
CARBOXIMID-DERIVATE ALS NÜTZLICHE UROSELEKTIVE ALPHA-1A ADRENOZEPTOR-BLOCKER
Title (fr)
DERIVES DE CARBOXIMIDE UTILES COMME BLOQUEURS UROSELECTIFS DU RECEPTEUR ADRENERGIQUE ALPHA-SB-1A
Publication
Application
Priority
IB 0201108 W 20020408
Abstract (en)
[origin: WO03084541A1] Novel carboximide derivatives, which selectively inhibit binding to the alpha >-1A< adrenergic receptor, a receptor which has been shown to be important in the treatment of benign prostatic hyperplasia. The compounds of the present invention are potentially useful in the treatment of benign prostatic hyperplasia.
IPC 1-7
IPC 8 full level
C07D 241/04 (2006.01); A61K 31/495 (2006.01); A61P 9/12 (2006.01); A61P 13/08 (2006.01); A61P 43/00 (2006.01); C07C 233/36 (2006.01); C07C 233/62 (2006.01); C07D 295/13 (2006.01)
CPC (source: EP)
A61P 9/12 (2017.12); A61P 13/08 (2017.12); A61P 43/00 (2017.12); C07D 295/13 (2013.01)
Citation (search report)
- [Y] WO 9737983 A1 19971016 - SOD CONSEILS RECH APPLIC [FR], et al
- [Y] WO 9906384 A1 19990211 - RECORDATI CHEM PHARM [CH], et al
- [DY] US 6083950 A 20000704 - ANAND NITYA [IN], et al
- See references of WO 03084541A1
Designated contracting state (EPC)
AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR
DOCDB simple family (publication)
WO 03084541 A1 20031016; AU 2002251409 A1 20031020; BR 0215686 A 20050222; CN 1627946 A 20050615; EA 200401335 A1 20060224; EP 1494674 A1 20050112; EP 1494674 A4 20060412; JP 2005532282 A 20051027; MX PA04009821 A 20041213
DOCDB simple family (application)
IB 0201108 W 20020408; AU 2002251409 A 20020408; BR 0215686 A 20020408; CN 02829097 A 20020408; EA 200401335 A 20020408; EP 02720343 A 20020408; JP 2003581781 A 20020408; MX PA04009821 A 20020408