Global Patent Index - EP 1572724 A4

EP 1572724 A4 20070314 - KDR AND VEGF/KDR BINDING PEPTIDES AND THEIR USE IN DIAGNOSIS AND THERAPY

Title (en)

KDR AND VEGF/KDR BINDING PEPTIDES AND THEIR USE IN DIAGNOSIS AND THERAPY

Title (de)

KDR UND VEGF/KDR BINDUNGSPEPTIDE UND IHRE VERWENDUNG BEI DER DIAGNOSE UND THERAPIE

Title (fr)

PEPTIDES LIANT DES RECEPTEURS KDR ET VEGF/KDR ET LEURS UTILISATIONS EN DIAGNOSTIC ET THERAPIE

Publication

EP 1572724 A4 20070314 (EN)

Application

EP 03711418 A 20030303

Priority

  • US 0306731 W 20030303
  • US 36085102 P 20020301
  • US 44041103 P 20030115

Abstract (en)

[origin: WO03074005A2] The present invention provides binding polypetides for KDR or VEGF/KDR complex, which have a variety of uses wherever treating, Detecting, isolating or localizing angiogenesis is advantageous. Particularly disclosed are synthetic, isolated polypeptides capable of binding KDR or VEGF/KDR complex with high affinity (e.g., having a KD<1 microM).

IPC 1-7

C07K 7/00

IPC 8 full level

A61K 49/22 (2006.01); A61K 51/08 (2006.01); C07K 7/08 (2006.01); C07K 14/00 (2006.01); C07K 14/52 (2006.01); C07K 14/71 (2006.01); A61K 38/00 (2006.01)

CPC (source: EP)

A61K 49/223 (2013.01); A61K 51/088 (2013.01); A61P 9/00 (2017.12); A61P 9/10 (2017.12); A61P 17/06 (2017.12); A61P 19/02 (2017.12); A61P 31/12 (2017.12); A61P 31/18 (2017.12); A61P 33/06 (2017.12); A61P 35/00 (2017.12); C07K 7/08 (2013.01); C07K 14/001 (2013.01); C07K 14/52 (2013.01); C07K 14/71 (2013.01); A61K 38/00 (2013.01); C07K 2319/00 (2013.01); Y02A 50/30 (2017.12)

Citation (search report)

  • [X] WO 0152875 A1 20010726 - LUDWIG INST CANCER RES [US]
  • [X] WO 0063380 A1 20001026 - GENENTECH INC [US]
  • [X] WO 0216412 A2 20020228 - DYAX CORP [US]
  • [X] HAIYAN JIA ET AL: "PEPTIDES ENCODED BY EXON 6 OF VEGF INHIBIT ENDOTHELIAL CELL BIOLOGICAL RESPONSES AND ANGIOGENESIS INDUCED BY VEGF", BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, ACADEMIC PRESS INC. ORLANDO, FL, US, vol. 283, no. 1, 2001, pages 164 - 173, XP002941058, ISSN: 0006-291X
  • [A] BINETRUY-TOURNAIRE ROSELYNE ET AL: "Identification of a peptide blocking vascular endothelial growth factor (VEGF)-mediated angiogenesis", EMBO JOURNAL, OXFORD UNIVERSITY PRESS, SURREY, GB, vol. 19, no. 7, 3 April 2000 (2000-04-03), pages 1525 - 1533, XP002179245, ISSN: 0261-4189
  • [A] SATO A K ET AL: "Development of mammalian serum albumin affinity purification media by peptide phage display", BIOTECHNOLOGY PROGRESS, XX, XX, vol. 18, no. 2, January 2002 (2002-01-01), pages 182 - 192, XP002348553, ISSN: 8756-7938
  • [A] FAIRBROTHER W J ET AL: "NOVEL PEPTIDES SELECTED TO BIND VASCULAR ENDOTHELIAL GROWTH FACTOR TARGET THE RECEPTOR-BINDING SITE", BIOCHEMISTRY, AMERICAN CHEMICAL SOCIETY. EASTON, PA, US, vol. 37, no. 51, 22 December 1998 (1998-12-22), pages 17754 - 17764, XP000876734, ISSN: 0006-2960
  • [T] SHRIVASTAVA A ET AL: "A distinct strategy to generate high-affinity peptide binders to receptor tyrosine kinases.", PROTEIN ENGINEERING, DESIGN & SELECTION : PEDS. SEP 2005, vol. 18, no. 9, September 2005 (2005-09-01), pages 417 - 424, XP002375785, ISSN: 1741-0126
  • [X] IWAMOTO Y ET AL: "YIGSR, A SYNTHETIC LAMININ PENTAPEPTIDE, INHIBITS EXPERIMENTAL METASTATIS FORMATION", SCIENCE, AMERICAN ASSOCIATION FOR THE ADVANCEMENT OF SCIENCE, US, vol. 238, no. 4830, 20 November 1987 (1987-11-20), pages 1132 - 1134, XP001135169, ISSN: 0036-8075
  • [X] LECOUTER JENNIFER ET AL: "Identification of an angiogenic mitogen selective for endocrine gland endothelium", NATURE, NATURE PUBLISHING GROUP, LONDON, GB, vol. 412, no. 6850, 30 August 2001 (2001-08-30), pages 877 - 884, XP002194811, ISSN: 0028-0836
  • See references of WO 03074005A2

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR

DOCDB simple family (publication)

WO 03074005 A2 20030912; WO 03074005 A8 20050721; AU 2003213730 A1 20030916; AU 2009201114 A1 20090409; AU 2009201114 B2 20120119; CA 2477836 A1 20030912; CA 2666005 A1 20030912; CA 2666005 C 20160119; EP 1572724 A2 20050914; EP 1572724 A4 20070314; EP 2014310 A2 20090114; EP 2014310 A3 20090909; EP 2014310 B1 20121024; EP 2014310 B8 20121226; EP 2301587 A2 20110330; EP 2301587 A3 20110406; EP 2301587 B1 20140625; ES 2398393 T3 20130315; ES 2506142 T3 20141013; JP 2006514915 A 20060518; JP 2009161549 A 20090723; JP 5039075 B2 20121003; SI 2301587 T1 20141128

DOCDB simple family (application)

US 0306731 W 20030303; AU 2003213730 A 20030303; AU 2009201114 A 20090319; CA 2477836 A 20030303; CA 2666005 A 20030303; EP 03711418 A 20030303; EP 08008365 A 20030303; EP 10185498 A 20030303; ES 08008365 T 20030303; ES 10185498 T 20030303; JP 2003572527 A 20030303; JP 2009049512 A 20090303; SI 200332390 T 20030303