Global Patent Index - EP 1581261 A4

EP 1581261 A4 20091021 - CYTOTOXINS AND DIAGNOSTIC IMAGING AGENTS COMPRISING HSP90 LIGANDS

Title (en)

CYTOTOXINS AND DIAGNOSTIC IMAGING AGENTS COMPRISING HSP90 LIGANDS

Title (de)

ZYTOTOXINE UND MITTEL FÜR DIAGNOSTISCHE BILDGEBUNG MIT HSP90-LIGANDEN

Title (fr)

CYTOTOXINES ET AGENTS D'IMAGERIE DE DIAGNOSTIC COMPRENANT DES LIGANDS HSP90

Publication

EP 1581261 A4 20091021 (EN)

Application

EP 03741983 A 20030612

Priority

  • US 0318776 W 20030612
  • US 0239993 W 20021212

Abstract (en)

[origin: WO2004054624A1] Cytotoxic compounds and diagnostic imaging agents comprising HSP90-ligands and methods of use thereof are described.

IPC 1-7

A61K 51/00; A61M 36/14; A61P 43/00

IPC 8 full level

C07D 225/06 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01); C07D 405/12 (2006.01); C07D 409/12 (2006.01); C07D 413/12 (2006.01); C07D 417/12 (2006.01); C07F 9/553 (2006.01)

CPC (source: EP)

A61K 47/54 (2017.07); A61K 51/04 (2013.01); A61P 43/00 (2017.12); C07D 225/06 (2013.01); C07D 401/12 (2013.01); C07D 403/12 (2013.01); C07D 405/12 (2013.01); C07D 409/12 (2013.01); C07D 413/12 (2013.01); C07D 417/12 (2013.01); C07F 9/5535 (2013.01)

Citation (search report)

  • [X] WO 0003737 A2 20000127 - US HEALTH [US], et al
  • [PX] WO 03045319 A2 20030605 - ACTIVBIOTICS INC [US], et al & ABSTRACTS OF PAPERS AMERICAN CHEMICAL SOCIETY, vol. 224, no. 1-2, 2002, 224TH NATIONAL MEETING OF THE AMERICAN CHEMICAL SOCIETY; BOSTON, MA, USA; AUGUST 18-22, 2002, pages BIOT 64, ISSN: 0065-7727
  • [X] DATABASE BIOSIS [online] BIOSCIENCES INFORMATION SERVICE, PHILADELPHIA, PA, US; 2002, MANDLER RAYA ET AL: "Strategies in conjugating geldanamycin derivatives to monoclonal antibodies that enhance herceptin efficacy in mice bearing HER2-overexpressing xenografts", XP002542020, Database accession no. PREV200200490291
  • [X] MANDLER R ET AL: "Synthesis and evaluation of antiproliferative activity of a geldanamycin-Herceptin TM immunoconjugate", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 10, no. 10, 1 May 2000 (2000-05-01), PERGAMON, ELSEVIER SCIENCE, GB, pages 1025 - 1028, XP004204597, ISSN: 0960-894X
  • [X] SCHNUR R C ET AL: "Preparation of 17-amino-22-(4'-azido-3'-<125>iodophenacyl)-17- demethoxygeldanamycin (1): An ansamycin for photoaffinity labeling", JOURNAL OF LABELLED COMPOUNDS AND RADIOPHARMACEUTICALS, vol. 34, no. 6, 1994, GB, pages 529 - 536, XP002542021, ISSN: 0362-4803
  • [X] FUKAZAWA H ET AL: "Labeling of v-Src and BCR-ABL tyrosine kinases with [<14>C]herbimycin A and its use in the elucidation of the kinase inactivation mechanism", FEBS LETTERS, vol. 340, no. 3, 1994, NL, pages 155 - 158, XP002542022, ISSN: 0014-5793
  • [DX] CHIOSIS GABRIELA ET AL: "A small molecule designed to bind to the adenine nucleotide pocket of Hsp90 causes Her2 degradation and the growth arrest and differentiation of breast cancer cells", CHEMISTRY AND BIOLOGY, vol. 8, no. 3, March 2001 (2001-03-01), LONDON, pages 289 - 299, XP002542023, ISSN: 1074-5521
  • See references of WO 2004054624A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR

DOCDB simple family (publication)

WO 2004054624 A1 20040701; AU 2003303058 A1 20040709; CA 2549463 A1 20040701; EP 1581261 A1 20051005; EP 1581261 A4 20091021

DOCDB simple family (application)

US 0318776 W 20030612; AU 2003303058 A 20030612; CA 2549463 A 20030612; EP 03741983 A 20030612