EP 1581478 A1 20051005 - DHODH-INHIBITORS AND METHOD FOR THEIR IDENTIFICATION
Title (en)
DHODH-INHIBITORS AND METHOD FOR THEIR IDENTIFICATION
Title (de)
DHODH-INHIBITOREN UND VERFAHREN ZU DEREN IDENTIFIKATION
Title (fr)
INHIBITEURS DE L'ENZYME DHODH ET LEUR PROCEDE D'IDENTIFICATION
Publication
Application
Priority
- EP 03813575 A 20031217
- DE 10260799 A 20021223
- DE 10260800 A 20021223
- EP 0314435 W 20031217
- EP 03028137 A 20031205
Abstract (en)
[origin: WO2004056747A1] The present invention relates to compounds of the general formula (I), or salts or isomeres thereof, wherein A is a 4-8 membered non-aromatic ring system, to compounds of the general formula (II), or salts or isomeres thereof, wherein A is a 3-8 membered non-aromatic ring system, wherein, when r = 0, there is no double bond between the carbon atoms carrying the substituents -CZ<1>- and -CZ<2>-;and to compounds of formula (III), wherein A is a heteroaromatic 5-membered ring system, which are capable of binding to the ubiquinone binding site of DHODH.
IPC 1-7
C07C 233/57; A61P 35/00; A61P 37/02; A61P 29/00; A61P 31/12; A61K 31/194; C07C 233/60; C07D 333/40; C07D 307/68; C07D 491/04; C07D 495/04; C07D 239/70; C07D 221/04; C07D 237/26
IPC 8 full level
A61K 31/194 (2006.01); A61P 29/00 (2006.01); A61P 31/12 (2006.01); A61P 35/00 (2006.01); A61P 37/02 (2006.01); C07C 233/57 (2006.01); C07C 233/60 (2006.01); C07C 235/40 (2006.01); C07C 235/82 (2006.01); C07D 221/04 (2006.01); C07D 237/26 (2006.01); C07D 239/70 (2006.01); C07D 307/68 (2006.01); C07D 333/38 (2006.01); C07D 333/40 (2006.01); C07D 491/04 (2006.01); C07D 495/04 (2006.01)
CPC (source: EP)
A61P 29/00 (2017.12); A61P 31/12 (2017.12); A61P 35/00 (2017.12); A61P 37/02 (2017.12); C07C 233/60 (2013.01); C07C 235/40 (2013.01); C07D 221/04 (2013.01); C07D 237/26 (2013.01); C07D 239/70 (2013.01); C07D 257/04 (2013.01); C07D 307/68 (2013.01); C07D 333/38 (2013.01); C07D 491/04 (2013.01); C07D 495/04 (2013.01); C07C 2601/08 (2017.04); C07C 2601/10 (2017.04)
Citation (search report)
See references of WO 2004056747A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PT RO SE SI SK TR
Designated extension state (EPC)
AL LT LV MK
DOCDB simple family (publication)
WO 2004056747 A1 20040708; AU 2003300530 A1 20040714; EP 1581478 A1 20051005
DOCDB simple family (application)
EP 0314435 W 20031217; AU 2003300530 A 20031217; EP 03813575 A 20031217