EP 1601669 A1 20051207 - SUBSTITUTED AZETIDINONE COMPOUNDS, FORMULATIONS AND USES THEREOF FOR THE TREATMENT OF HYPERCHOLESTEROLEMIA
Title (en)
SUBSTITUTED AZETIDINONE COMPOUNDS, FORMULATIONS AND USES THEREOF FOR THE TREATMENT OF HYPERCHOLESTEROLEMIA
Title (de)
SUBSTITUIERTE AZETIDINON-DERIVATE, DEREN PHARMAZEUTISCHE FORMULIERUNGEN UND DEREN VERWENDUNG ZUR BEHANDLUNG VON HYPERCHOLESTEROLEMIA
Title (fr)
COMPOSES D'AZETIDINONE SUBSTITUES, LEURS FORMULATIONS ET LEUR UTILISATION POUR TRAITER L'HYPERCHOLESTEROLEMIE
Publication
Application
Priority
- US 2004006428 W 20040303
- US 45272503 P 20030307
Abstract (en)
[origin: US7732413B2] The present invention provides compounds represented by the structural formula (I): or pharmaceutically acceptable isomers, salts, solvates or esters of the compound of Formula (I), wherein each of the substituents is as specified herein, formulations including the above compounds, processes for preparing the same and methods for treating atherosclerosis, hypercholesterolemia, or sitosterolemia, and for lowering plasma levels of sterols and/or stanols.
IPC 1-7
IPC 8 full level
A61P 3/06 (2006.01); C07D 405/12 (2006.01); C07D 405/14 (2006.01)
CPC (source: EP US)
A61P 3/04 (2018.01 - EP); A61P 3/06 (2018.01 - EP); A61P 3/10 (2018.01 - EP); A61P 9/00 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 25/00 (2018.01 - EP); A61P 25/28 (2018.01 - EP); A61P 43/00 (2018.01 - EP); C07D 405/12 (2013.01 - EP US); C07D 405/14 (2013.01 - EP US); Y10S 930/28 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
US 2004180861 A1 20040916; US 7208486 B2 20070424; AT E418551 T1 20090115; CA 2517572 A1 20040923; CA 2517572 C 20111213; CN 1756756 A 20060405; DE 602004018617 D1 20090205; EP 1601669 A1 20051207; EP 1601669 B1 20081224; ES 2318274 T3 20090501; HK 1085728 A1 20060901; JP 2007524597 A 20070830; JP 2010254719 A 20101111; JP 4589919 B2 20101201; MX PA05009501 A 20051018; US 2007155676 A1 20070705; US 2008200446 A1 20080821; US 7378518 B2 20080527; US 7732413 B2 20100608; WO 2004081003 A1 20040923
DOCDB simple family (application)
US 79234604 A 20040303; AT 04716913 T 20040303; CA 2517572 A 20040303; CN 200480006048 A 20040303; DE 602004018617 T 20040303; EP 04716913 A 20040303; ES 04716913 T 20040303; HK 06105698 A 20060516; JP 2006509018 A 20040303; JP 2010181957 A 20100816; MX PA05009501 A 20040303; US 10872908 A 20080424; US 2004006428 W 20040303; US 70844907 A 20070220