EP 1603535 A4 20081015 - AROMATASE INHIBITOR DIAGNOSIS AND THERAPY
Title (en)
AROMATASE INHIBITOR DIAGNOSIS AND THERAPY
Title (de)
AROMATASE-HEMMER-DIAGNOSE UND THERAPIE
Title (fr)
DIAGNOSTIC ET TRAITEMENT FAISANT APPEL A UN INHIBITEUR DE L'AROMATASE
Publication
Application
Priority
- US 2004008082 W 20040317
- US 45551003 P 20030318
Abstract (en)
[origin: WO2004082626A2] The present invention provides pharmaceutical compositions which are useful for imaging and/or treating endometriosis. The compositions are useful for the treatment of reproductive age women, as well as post-menopausal women suffering from this disorder. The pharmaceutical composition is a liposome composition that includes a liposome carrier component that contains on its surface a moiety targeted for an endometriotic implant or leaky blood vessels within the implant. The inventive liposome composition includes an aromatase inhibitor and/or a radiolabeled complex encapsulated by the liposome component. A label capable of external detection can be included so as to permit the detection of an endometrial implant and/or diagnosis of the presence of endornetriosis in a patient. The label can be bound to the aromatase inhibitor. Alternatively, when the label is separate from the inhibitor, or when the inhibitor is not present, a radiolabeled complex can be included.
IPC 8 full level
A61K 9/127 (2006.01); A61K 9/133 (2006.01); A61K 51/12 (2006.01); A61P 15/00 (2006.01)
IPC 8 main group level
A61K (2006.01)
CPC (source: EP)
A61K 9/1271 (2013.01); A61K 9/1272 (2013.01); A61K 51/1234 (2013.01); A61P 15/00 (2017.12)
Citation (search report)
- [X] WO 0193836 A2 20011213 - BOULIKAS TENI [US]
- [X] WO 0062813 A2 20001026 - UNIV BRITISH COLUMBIA [CA], et al
- [Y] WO 0120990 A1 20010329 - BIORESPONSE LLC [US]
- [A] WO 02096927 A2 20021205 - RIBOZYME PHARM INC [US], et al
- [A] US 2002177574 A1 20021128 - TAYLOR HUGH S [US]
- [Y] TAKAYAMA KAZUTO ET AL: "Treatment of severe postmenopausal endometriosis with an aromatase inhibitor", FERTILITY AND STERILITY, ELSEVIER SCIENCE INC, NEW YORK, NY, US, vol. 69, no. 4, 1 April 1998 (1998-04-01), pages 709 - 713, XP002379276, ISSN: 0015-0282
- See references of WO 2004082626A2
Designated contracting state (EPC)
DE ES FR GB IT
DOCDB simple family (publication)
WO 2004082626 A2 20040930; WO 2004082626 A3 20041111; EP 1603535 A2 20051214; EP 1603535 A4 20081015
DOCDB simple family (application)
US 2004008082 W 20040317; EP 04757537 A 20040317