EP 1660454 A1 20060531 - AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS
Title (en)
AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS
Title (de)
AZAZYKLISCHE VERBINDUNGEN ALS INHIBITOREN VON SNS (SENSORY NEURONE SPECIFIC)-KANALEN
Title (fr)
COMPOSES AZACYCLIQUES CONVENANT COMME INHIBITEURS DES CANAUX SPECIFIQUES DES NEURONES SENSORIELS
Publication
Application
Priority
- GB 2004002945 W 20040707
- GB 0315872 A 20030707
- US 48844203 P 20030721
Abstract (en)
[origin: WO2005005392A1] Compounds of the formula (I), and pharmaceutically acceptable salts thereof, are found to be antagonists of SNS sodium channels. They are therefore useful as analgesic and neuroprotective agents wherein: X is -N- or -CH-; n is from 0 to 3.
IPC 1-7
C07D 217/04; C07D 209/44; C07D 403/06; C07D 223/16; A61K 31/472; A61K 31/4035; A61K 31/55; A61P 25/04
IPC 8 full level
A61P 25/04 (2006.01); C07D 209/44 (2006.01); C07D 209/86 (2006.01); C07D 217/02 (2006.01); C07D 217/10 (2006.01); C07D 217/14 (2006.01); C07D 217/22 (2006.01); C07D 223/16 (2006.01); C07D 401/06 (2006.01); C07D 401/12 (2006.01); C07D 403/06 (2006.01); C07D 409/06 (2006.01); C07D 413/06 (2006.01); C07D 413/12 (2006.01); C07D 417/06 (2006.01); C07D 417/12 (2006.01); C07D 471/04 (2006.01); C07D 487/04 (2006.01)
CPC (source: EP)
A61P 25/04 (2018.01); C07D 209/44 (2013.01); C07D 209/86 (2013.01); C07D 217/02 (2013.01); C07D 217/10 (2013.01); C07D 217/14 (2013.01); C07D 217/22 (2013.01); C07D 223/16 (2013.01); C07D 401/06 (2013.01); C07D 401/12 (2013.01); C07D 403/06 (2013.01); C07D 409/06 (2013.01); C07D 413/06 (2013.01); C07D 413/12 (2013.01); C07D 417/06 (2013.01); C07D 417/12 (2013.01); C07D 471/04 (2013.01); C07D 487/04 (2013.01)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
DOCDB simple family (application)
GB 2004002945 W 20040707; EP 04743288 A 20040707