EP 1667679 B1 20090603 - AMINOBENZIMIDAZOLES AS SELECTIVE MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF OBESITY AND RELATED DISORDERS
Title (en)
AMINOBENZIMIDAZOLES AS SELECTIVE MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF OBESITY AND RELATED DISORDERS
Title (de)
AMINOBENZIMIDAZOLE ALS SELEKTIVE MELANIN-KONZENTRIERENDE HORMON-REZEPTORANTAGONISTEN ZUR BEHANDLUNG VON FETTSUCHT UND VERWANDTEN ERKRANKUNGEN
Title (fr)
AMINOBENZIMIDAZOLES UTILISES EN TANT QU'ANTAGONISTES SELECTIFS DES RECEPTEURS DE L'HORMONE CONCENTRANT LA MELANINE (MCH) POUR LE TRAITEMENT DE L'OBESITE ET DES TROUBLES ASSOCIES
Publication
Application
Priority
- US 2004032494 W 20040930
- US 50802703 P 20031002
Abstract (en)
[origin: WO2005034947A1] The present invention discloses compounds of formula I formula I wherein Ar, Z, m, n, p, R<1> and R<8> are herein defined, said compounds being novel antagonists for melanin-concentrating hormone (MCH), as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising such MCH antagonists as well as methods of using them to treat obesity, metabolic disorders, eating disorders such as hyperphagia, and diabetes.
IPC 8 full level
A61K 31/4184 (2006.01); A61P 3/04 (2006.01); C07D 235/30 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01)
CPC (source: EP US)
A61P 3/00 (2018.01 - EP); A61P 3/04 (2018.01 - EP); A61P 3/06 (2018.01 - EP); A61P 3/10 (2018.01 - EP); A61P 9/12 (2018.01 - EP); C04B 35/632 (2013.01 - EP US); C07D 235/30 (2013.01 - EP US); C07D 401/12 (2013.01 - EP US); C07D 403/12 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR
Designated extension state (EPC)
AL HR LT LV MK
DOCDB simple family (publication)
WO 2005034947 A1 20050421; AT E432702 T1 20090615; CA 2540845 A1 20050421; CA 2540845 C 20101109; CN 1859907 A 20061108; DE 602004021399 D1 20090716; EP 1667679 A1 20060614; EP 1667679 B1 20090603; ES 2326980 T3 20091022; JP 2007507533 A 20070329; MX PA06003738 A 20060614; US 2005085488 A1 20050421; US 7030113 B2 20060418
DOCDB simple family (application)
US 2004032494 W 20040930; AT 04789487 T 20040930; CA 2540845 A 20040930; CN 200480028600 A 20040930; DE 602004021399 T 20040930; EP 04789487 A 20040930; ES 04789487 T 20040930; JP 2006534183 A 20040930; MX PA06003738 A 20040930; US 95478604 A 20040930