EP 1689408 A4 20100303 - TREATMENT OF INFLAMMATORY DISORDERS OF THE EPITHELIUM WITH LOW DOSE 2,3-BENZODIAZEPINES
Title (en)
TREATMENT OF INFLAMMATORY DISORDERS OF THE EPITHELIUM WITH LOW DOSE 2,3-BENZODIAZEPINES
Title (de)
BEHANDLUNG VON ENTZÜNDLICHEN ERKRANKUNGEN DES EPITHELS MIT NIEDRIGDOSIERTEN 2,3-BENZODIAZEPINEN
Title (fr)
TRAITEMENT DE TROUBLES INFLAMMATOIRES DE L'EPITHELIUM AU MOYEN DE 2,3-BENZODIAZEPINES EN FAIBLE DOSE
Publication
Application
Priority
- US 2004040403 W 20041203
- US 0338643 W 20031203
- US 72794003 A 20031203
Abstract (en)
[origin: WO2005056017A1] Compounds according to formula (I) wherein R<1>, R<2>, R<3>, R<4>, R<5> and n are as defined herein, are administered at low dosage for the prevention or treatment of inflammatory disorders, particularly those affecting epithelial tissues such as those of the skin and gastrointestinal tract.
IPC 8 full level
A61K 31/55 (2006.01); A61K 31/551 (2006.01); A61P 1/00 (2006.01); A61P 17/00 (2006.01); A61P 29/00 (2006.01)
CPC (source: EP)
A61K 31/55 (2013.01); A61K 31/551 (2013.01); A61P 1/00 (2017.12); A61P 1/02 (2017.12); A61P 1/04 (2017.12); A61P 17/00 (2017.12); A61P 17/06 (2017.12); A61P 19/06 (2017.12); A61P 27/02 (2017.12); A61P 29/00 (2017.12)
Citation (search report)
- [PX] WO 2004050080 A1 20040617 - VELA PHARMACEUTICALS INC [US], et al
- [X] YOSHIKAWA K ET AL: "Clinical evaluation of Grandaxin(R) (tofisopam) on several skin diseases", SKIN RESEARCH 1993 JP, vol. 35, no. 1, 1993, pages 195 - 202, XP009128520, ISSN: 0018-1390
- [X] KONO T ET AL: "CLINICAL EVALUATION OF TOFISOPAM GRANDAXIN ON SEVERAL DERMATOLOGICAL DISEASES IN PATIENTS WITH PSYCHOSOMATIC SYMPTOMS", HIFU, vol. 33, no. 6, 1991, pages 699 - 707, XP009128521, ISSN: 0018-1390
- [PX] LEVENTER STEVEN M ET AL: "The potential of dextofisopam for treatment of irritable bowel syndrome and inflammatory bowel disease", AMERICAN JOURNAL OF GASTROENTEROLOGY, vol. 99, no. 10, Suppl. S, October 2004 (2004-10-01), & 69TH ANNUAL MEETING OF THE AMERICAN-COLLEGE-OF-GASTROENTEROLOGY; ORLANDO, FL, USA; OCTOBER 29 -NOVEMBER 03, 2004, pages S279, XP009128474, ISSN: 0002-9270
- See references of WO 2005056017A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2005056017 A1 20050623; CA 2548038 A1 20050623; EP 1689408 A1 20060816; EP 1689408 A4 20100303; JP 2007513171 A 20070524
DOCDB simple family (application)
US 2004040403 W 20041203; CA 2548038 A 20041203; EP 04812836 A 20041203; JP 2006542754 A 20041203