EP 1689439 A2 20060816 - SMALL MOLECULE COMPOSITIONS AND METHODS FOR INCREASING DRUG EFFICIENCY USING COMPOSITIONS THEREOF
Title (en)
SMALL MOLECULE COMPOSITIONS AND METHODS FOR INCREASING DRUG EFFICIENCY USING COMPOSITIONS THEREOF
Title (de)
KLEINMOLEKÜLIGE ZUSAMMENSETZUNGEN UND VERFAHREN ZUR ERHÖHUNG DER ARZNEIMITTELEFFIZIENZ UNTER VERWENDUNG VON ZUSAMMENSETZUNGEN DAVON
Title (fr)
COMPOSITIONS A PETITES MOLECULES ET PROCEDES DESTINES A AUGMENTER L'EFFICACITE D'UN MEDICAMENT AU MOYEN DE CES COMPOSITIONS
Publication
Application
Priority
- US 2004031147 W 20040922
- US 50532503 P 20030922
- US 58183504 P 20040622
Abstract (en)
[origin: WO2005030258A2] In certain embodiments, provided herein are compositions and methods for increasing drug efficiency. The conjugates provided are in certain embodiments, for compositions and methods in treatment of variety of diseases and have the formula 1: D - L - S (1) or formula 2: D-L-S' (2) wherein D is a drug moiety; L, which may or may not be present, is a non-releasing linker moiety; S is a substrate for a kinase, other than a hexokinase, a protein kinase or a lipid kinase; and S' is a substrate for a phosphotransferase, other than a hexokinase, a protein kinase or a lipid kinase.
IPC 8 full level
A61K 47/48 (2006.01); A61K 31/337 (2006.01); A61K 31/475 (2006.01); A61K 31/704 (2006.01); A61K 49/04 (2006.01); C07H 21/00 (2006.01); C07K 7/08 (2006.01); A61K 38/00 (2006.01)
CPC (source: EP)
A61K 31/337 (2013.01); A61K 31/475 (2013.01); A61K 31/704 (2013.01); A61K 49/0404 (2013.01); A61P 9/10 (2017.12); A61P 11/06 (2017.12); A61P 13/12 (2017.12); A61P 17/00 (2017.12); A61P 17/06 (2017.12); A61P 19/02 (2017.12); A61P 19/10 (2017.12); A61P 25/00 (2017.12); A61P 27/02 (2017.12); A61P 29/00 (2017.12); A61P 35/00 (2017.12); A61P 35/02 (2017.12); A61P 35/04 (2017.12); A61P 37/02 (2017.12); A61P 37/06 (2017.12); A61P 43/00 (2017.12); C07K 7/08 (2013.01); A61K 38/00 (2013.01)
Citation (search report)
See references of WO 2005030258A2
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IT LI LU MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2005030258 A2 20050407; WO 2005030258 A3 20050922; AU 2004275770 A1 20050407; CA 2539914 A1 20050407; EP 1689439 A2 20060816; JP 2007522094 A 20070809
DOCDB simple family (application)
US 2004031147 W 20040922; AU 2004275770 A 20040922; CA 2539914 A 20040922; EP 04784836 A 20040922; JP 2006527154 A 20040922