Global Patent Index - EP 1720885 A1

EP 1720885 A1 20061115 - A PROCESS FOR MAKING OLANZAPINE IN A POLYMORPH FORM I

Title (en)

A PROCESS FOR MAKING OLANZAPINE IN A POLYMORPH FORM I

Title (de)

VERFAHREN ZUR HERSTELLUNG VON OLANZAPIN IN EINER POLYMORPHEN FORM I

Title (fr)

PROCEDE DE FABRICATION D'OLANZAPINE SOUS FORME POLYMORPHE I

Publication

EP 1720885 A1 20061115 (EN)

Application

EP 05701231 A 20050126

Priority

  • EP 2005000834 W 20050126
  • US 53912004 P 20040127
  • US 56222504 P 20040415
  • US 56960704 P 20040511

Abstract (en)

[origin: WO2005070937A1] Heating a solid, preferably crystalline, olanzapine acetate can produce olanzapine Form I in high purity, free of other olanzapine forms and in good yields. The olanzapine acetate can also be used to purify raw or technical grade olanzapine and to serve as an intermediary to other forms of olanzapine base.

IPC 8 full level

C07D 495/04 (2006.01); A61K 31/55 (2006.01)

CPC (source: EP)

C07D 495/04 (2013.01)

Citation (search report)

See references of WO 2005070937A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC NL PL PT RO SE SI SK TR

DOCDB simple family (publication)

WO 2005070937 A1 20050804; AR 047460 A1 20060118; AR 047461 A1 20060118; EP 1711503 A1 20061018; EP 1720885 A1 20061115; WO 2005070939 A1 20050804

DOCDB simple family (application)

EP 2005000834 W 20050126; AR P050100259 A 20050126; AR P050100260 A 20050126; EP 05701231 A 20050126; EP 05707056 A 20050126; EP 2005000836 W 20050126