Global Patent Index - EP 1737864 A1

EP 1737864 A1 20070103 - SELECTED CGRP ANTAGONISTS, METHODS FOR THE PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS

Title (en)

SELECTED CGRP ANTAGONISTS, METHODS FOR THE PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS

Title (de)

AUSGEWAEHLTE CGRP-ANTAGONISTEN, VERFAHREN ZU DEREN HERSTELLUNG SOWIE DEREN VERWENDUNG ALS ARZNEIMITTEL

Title (fr)

ANTAGONISTES DU CGRP SELECTIONNES, LEURS PROCEDES DE PRODUCTION ET LEUR UTILISATION COMME MEDICAMENT

Publication

EP 1737864 A1 20070103 (DE)

Application

EP 05731903 A 20050412

Priority

  • EP 2005003816 W 20050412
  • DE 102004018794 A 20040415

Abstract (en)

[origin: WO2005100360A1] The invention relates to the CGRP antagonists of general formula (I), wherein A and R<1> to R<3> are defined as indicated in claim 1, the tautomers, diastereomers, enantiomers, hydrates, mixtures and salts thereof, the hydrates of the salts, especially the physiologically acceptable salts thereof with inorganic or organic acids, medicaments containing said compounds, the use thereof, and methods for the production thereof.

IPC 8 full level

C07D 471/10 (2006.01); A61K 31/438 (2006.01); A61K 31/527 (2006.01); A61K 31/537 (2006.01); A61P 3/10 (2006.01); A61P 25/06 (2006.01); C07D 498/10 (2006.01); C07D 519/00 (2006.01)

CPC (source: EP)

A61P 1/02 (2017.12); A61P 1/12 (2017.12); A61P 3/10 (2017.12); A61P 5/24 (2017.12); A61P 9/00 (2017.12); A61P 11/00 (2017.12); A61P 11/06 (2017.12); A61P 15/12 (2017.12); A61P 17/00 (2017.12); A61P 17/02 (2017.12); A61P 19/02 (2017.12); A61P 25/06 (2017.12); A61P 25/36 (2017.12); A61P 27/16 (2017.12); A61P 29/00 (2017.12); A61P 31/04 (2017.12); A61P 37/08 (2017.12); A61P 39/02 (2017.12); A61P 43/00 (2017.12); C07D 471/10 (2013.01)

Citation (search report)

See references of WO 2005100360A1

Citation (examination)

WERMUTH C.G.: "MOLECULAR VARIATIONS BASED ON ISOSTERIC REPLACEMENTS", PRACTICE OF MEDICINAL CHEMISTRY, 1996, pages 203 - 237, XP002190259

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC NL PL PT RO SE SI SK TR

Designated extension state (EPC)

BA HR YU

DOCDB simple family (publication)

WO 2005100360 A1 20051027; CA 2562529 A1 20051027; DE 102004018794 A1 20051027; EP 1737864 A1 20070103; JP 2007532602 A 20071115

DOCDB simple family (application)

EP 2005003816 W 20050412; CA 2562529 A 20050412; DE 102004018794 A 20040415; EP 05731903 A 20050412; JP 2007507731 A 20050412