Global Patent Index - EP 1757598 A4

EP 1757598 A4 20100721 - SUBSTITUTED PYRROLIDINE DERIVATIVE

Title (en)

SUBSTITUTED PYRROLIDINE DERIVATIVE

Title (de)

SUBSTITUIERTES PYRROLIDINDERIVAT

Title (fr)

DÉRIVÉ DE PYRROLIDINE SUBSTITUÉE

Publication

EP 1757598 A4 20100721 (EN)

Application

EP 05738631 A 20050513

Priority

  • JP 2005008750 W 20050513
  • JP 2004143352 A 20040513

Abstract (en)

[origin: EP1757598A1] The present invention contemplates provision of a quinolone antibacterial agent and a drug for the treatment of infectious diseases, which exhibit potent antibacterial activity and higher selective toxicity against Gram-positive and Gram-negative bacteria, which do not cause side effects (e.g., convulsion), and which exhibit higher safety. A compound represented by the following formula (I): a salt of the compound, or a hydrate of the compound or the salt; and an antibacterial drug and an infectious disease treating drug containing the compound as an active ingredient.

IPC 8 full level

A61K 31/4709 (2006.01); A61K 31/5383 (2006.01); A61P 31/04 (2006.01); C07D 401/04 (2006.01); C07D 498/06 (2006.01)

CPC (source: EP US)

A61P 31/00 (2017.12 - EP); A61P 31/04 (2017.12 - EP); C07D 401/04 (2013.01 - EP US); C07D 498/06 (2013.01 - EP US)

Citation (search report)

  • [X] EP 0208210 A1 19870114 - KYORIN SEIYAKU KK [JP]
  • [X] WO 03076428 A1 20030918 - DAIICHI SEIYAKU CO [JP], et al
  • [X] WO 03097634 A1 20031127 - DAIICHI SEIYAKU CO [JP], et al
  • [XP] WO 2004058261 A1 20040715 - DAIICHI SEIYAKU CO [JP], et al
  • [E] EP 1712554 A1 20061018 - DAIICHI SEIYAKU CO [JP]
  • [X] KAWAKAMI K ET AL: "Studies on 8-methoxyquinolones: synthesis and antibacterial activity of 7-(3-amino-4-substituted)pyrrolidinyl derivatives", 20001101, vol. 48, no. 11, 1 November 2000 (2000-11-01), pages 1667 - 1672, XP002989094
  • [X] K. KAWAKAMI ET AL.: "synthesis and antibacterial activity of novel pyridobenzoxazine", CHEMICAL AND PHARMACEUTICAL BULLETIN., vol. 46, no. 11, 1998, JPPHARMACEUTICAL SOCIETY OF JAPAN. TOKYO., pages 1710 - 1715, XP002586038, ISSN: 0009-2363
  • See references of WO 2005111015A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC NL PL PT RO SE SI SK TR

DOCDB simple family (publication)

EP 1757598 A1 20070228; EP 1757598 A4 20100721; JP 4820290 B2 20111124; JP WO2005111015 A1 20080321; US 2008045520 A1 20080221; US 2011166131 A1 20110707; US 7977327 B2 20110712; US 8455482 B2 20130604; WO 2005111015 A1 20051124

DOCDB simple family (application)

EP 05738631 A 20050513; JP 2005008750 W 20050513; JP 2006513559 A 20050513; US 201113045567 A 20110311; US 59631805 A 20050513