EP 1763516 A2 20070321 - SUBSTITUTED TETRAHYDROISOCHINOLINES USED IN THE FORM OF MMP INHIBITORS, METHOD FOR THE PRODUCTION AND USE THEREOF IN THE FORM OF DRAGS
Title (en)
SUBSTITUTED TETRAHYDROISOCHINOLINES USED IN THE FORM OF MMP INHIBITORS, METHOD FOR THE PRODUCTION AND USE THEREOF IN THE FORM OF DRAGS
Title (de)
SUBSTITUIERTE TETRAHYDROISOCHINOLINE ALS MMP-INHIBITOREN, VERFAHREN ZU IHRER HERSTELLUNG UND IHRE VERWENDUNG ALS MEDIKAMENT
Title (fr)
TETRAHYDRO-ISOQUINOLEINES SUBSTITUEES, UTILISEES COMME INHIBITEURS MMP, LEUR PROCEDE DE FABRICATION ET LEUR UTILISATION COMME MEDICAMENTS
Publication
Application
Priority
- EP 2005006415 W 20050615
- DE 102004031850 A 20040630
Abstract (en)
[origin: US2007203118A1] The present invention is directed to a compound of formula (I) wherein R<SUB>1</SUB>, R<SUB>2</SUB>, R<SUB>3</SUB>, R<SUB>4</SUB>, A, L and n are as defined herein, or a pharmacologically acceptable salt thereof, its pharmaceutical composition and it use as a MMP inhibitor.
IPC 8 full level
C07D 217/26 (2006.01); A61K 31/472 (2006.01); A61P 9/10 (2006.01); A61P 19/02 (2006.01); C07D 217/14 (2006.01)
CPC (source: EP KR US)
A61K 31/4035 (2013.01 - KR); A61K 31/472 (2013.01 - KR); A61P 1/02 (2017.12 - EP); A61P 1/04 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/04 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 17/02 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 19/04 (2017.12 - EP); A61P 19/10 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 217/14 (2013.01 - EP KR US); C07D 217/26 (2013.01 - EP KR US); C07D 401/12 (2013.01 - KR)
Citation (search report)
See references of WO 2006002763A2
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
US 2007203118 A1 20070830; AU 2005259633 A1 20060112; BR PI0511323 A 20071204; CA 2572125 A1 20060112; CN 101006059 A 20070725; DE 102004031850 A1 20060126; EP 1763516 A2 20070321; IL 179974 A0 20070515; JP 2008504315 A 20080214; KR 20070026679 A 20070308; MX PA06014366 A 20070308; PE 20060458 A1 20060529; TW 200612940 A 20060501; UY 28993 A1 20060131; WO 2006002763 A2 20060112; WO 2006002763 A3 20060316
DOCDB simple family (application)
US 61293806 A 20061219; AU 2005259633 A 20050615; BR PI0511323 A 20050615; CA 2572125 A 20050615; CN 200580022096 A 20050615; DE 102004031850 A 20040630; EP 05757350 A 20050615; EP 2005006415 W 20050615; IL 17997406 A 20061211; JP 2007518484 A 20050615; KR 20067027661 A 20061228; MX PA06014366 A 20050615; PE 2005000688 A 20050616; TW 94121519 A 20050628; UY 28993 A 20050630