EP 1778691 A1 20070502 - HYDRATES AND POLYMORPHS OF 4-[[(7R)-8-CYCLOPENTYL-7-ETHYL-5,6,7,8-TETRAHYDRO-5-METHYL-4-6-OXO-2-PIPERIDINYL]AMINO]-3-METHOXY-N-(1-METHYL-4-PIPERIDINYL)-BENZAMIDE, METHODS FOR THE PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS
Title (en)
HYDRATES AND POLYMORPHS OF 4-[[(7R)-8-CYCLOPENTYL-7-ETHYL-5,6,7,8-TETRAHYDRO-5-METHYL-4-6-OXO-2-PIPERIDINYL]AMINO]-3-METHOXY-N-(1-METHYL-4-PIPERIDINYL)-BENZAMIDE, METHODS FOR THE PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS
Title (de)
HYDRATE UND POLYMORPHE DES 4-[[(7R)-8-CYCLOPENTYL-7-ETHYL-5,6,7,8-TETRAHYDRO-5-METHYL-4-6-OXO-2-PIPERIDINYL ]AMINO]-3-METHOXY-N-(1-METHYL-4-PIPERIDINYL)-BENZAMID, VERFAHREN ZU DEREN HERSTELLUNG UND DEREN VERWENDUNG ALS ARZNEIMITTEL
Title (fr)
NOUVEAUX HYDRATES ET POLYMORPHES DU 4-[[(7R)-8-CYCLOPENTYL-7-ETHYL-5,6,7,8-TETRAHYDRO-5-METHYL-4-6-OXO-2-PIPERIDINYL]AMINO]-3-METHOXY-N-(1-METHYL-4-PIPERIDINYL)-BENZAMIDE, SON PROCEDE DE PRODUCTION ET SON UTILISATION COMME MEDICAMENT
Publication
Application
Priority
- EP 2005008736 W 20050811
- EP 04019366 A 20040814
- EP 05772062 A 20050811
Abstract (en)
[origin: US2006035902A1] Disclosed are hydrates and polymorphs of 4-[[(7R)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-6-oxo-2-pteridinyl]amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide, processes for preparing them and their use as pharmaceutical compositions.
IPC 8 full level
C07D 475/00 (2006.01); A61K 31/519 (2006.01); A61P 35/00 (2006.01); C07D 211/58 (2006.01)
CPC (source: EP KR US)
A61K 31/519 (2013.01 - KR); A61P 29/00 (2017.12 - EP); A61P 31/04 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 37/00 (2017.12 - EP); A61P 37/02 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 211/58 (2013.01 - EP US); C07D 475/00 (2013.01 - EP KR US)
Citation (search report)
See references of WO 2006018222A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
Designated extension state (EPC)
BA HR YU
DOCDB simple family (publication)
US 2006035902 A1 20060216; US 7728134 B2 20100601; AR 052404 A1 20070321; AU 2005274340 A1 20060223; AU 2005274340 B2 20120405; BR PI0514351 A2 20121030; CA 2578098 A1 20060223; CN 101006090 A 20070725; EA 011407 B1 20090227; EA 200700387 A1 20070831; EC SP077249 A 20070329; EP 1778691 A1 20070502; IL 181302 A0 20070704; JP 2008509953 A 20080403; KR 101221864 B1 20130114; KR 20070050967 A 20070516; MX 2007001854 A 20070328; NO 20070752 L 20070510; NZ 553649 A 20101126; PE 20060424 A1 20060609; TW 200619220 A 20060616; TW I370131 B 20120811; UA 87865 C2 20090825; US 2009298840 A1 20091203; US 2009318457 A1 20091224; US 8034816 B2 20111011; US 8202867 B2 20120619; WO 2006018222 A1 20060223; WO 2006018222 A8 20060615
DOCDB simple family (application)
US 19763405 A 20050804; AR P050103385 A 20050812; AU 2005274340 A 20050811; BR PI0514351 A 20050811; CA 2578098 A 20050811; CN 200580027683 A 20050811; EA 200700387 A 20050811; EC SP077249 A 20070214; EP 05772062 A 20050811; EP 2005008736 W 20050811; IL 18130207 A 20070213; JP 2007526360 A 20050811; KR 20077005956 A 20050811; MX 2007001854 A 20050811; NO 20070752 A 20070208; NZ 55364905 A 20050811; PE 2005000934 A 20050812; TW 94127602 A 20050812; UA A200702574 A 20050811; US 47817809 A 20090604; US 47818309 A 20090604