EP 1831194 A1 20070912 - HETEROCYCLIC MCHr1 ANTAGONISTS AND THEIR USE IN THERAPY
Title (en)
HETEROCYCLIC MCHr1 ANTAGONISTS AND THEIR USE IN THERAPY
Title (de)
HETEROCYCLISCHE MCHR1-ANTAGONISTEN UND DEREN VERWENDUNG IN DER THERAPIE
Title (fr)
ANTAGONISTES HETEROCYCLIQUES DE MCHr1 ET LEURS APPLICATIONS THERAPEUTIQUES
Publication
Application
Priority
- SE 2005001966 W 20051219
- SE 0403119 A 20041221
- SE 0501686 A 20050715
Abstract (en)
[origin: WO2006068594A1] Compounds of formula I depicted below, pharmaceutical compositions containing them, processes for preparing the compounds, and their use in the treatment of obesity, type II diabetes, metabolic syndrome, psychiatric disorders, cognitive disorders, memory disorders, schizophrenia, epilepsy and related conditions, neurological disorders such as dementia, multiple sclerosis, Parkinson's disease, Huntington's chorea and Alzheimer's disease, and pain related disorders. The compounds are melanin concentrating hormone receptor 1 (MCHr1) antagonists.
IPC 8 full level
C07D 401/06 (2006.01); A61K 31/4025 (2006.01); A61K 31/4427 (2006.01); A61K 31/4523 (2006.01); A61K 31/496 (2006.01); A61P 3/04 (2006.01); A61P 3/10 (2006.01); A61P 25/00 (2006.01); C07D 401/14 (2006.01); C07D 405/14 (2006.01); C07D 413/14 (2006.01); C07D 417/14 (2006.01)
CPC (source: EP US)
A61P 1/04 (2017.12 - EP); A61P 3/04 (2017.12 - EP); A61P 3/10 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 11/00 (2017.12 - EP); A61P 15/00 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/04 (2017.12 - EP); A61P 25/06 (2017.12 - EP); A61P 25/08 (2017.12 - EP); A61P 25/14 (2017.12 - EP); A61P 25/16 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 25/22 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 25/30 (2017.12 - EP); A61P 25/32 (2017.12 - EP); A61P 25/34 (2017.12 - EP); A61P 25/36 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 29/02 (2017.12 - EP); A61P 37/02 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 401/06 (2013.01 - EP US); C07D 401/12 (2013.01 - EP US); C07D 401/14 (2013.01 - EP US); C07D 405/14 (2013.01 - EP US); C07D 413/14 (2013.01 - EP US); C07D 417/14 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2006068594 A1 20060629; AR 051802 A1 20070207; EP 1831194 A1 20070912; EP 1831194 A4 20091202; JP 2008524325 A 20080710; TW 200635589 A 20061016; US 2008306055 A1 20081211
DOCDB simple family (application)
SE 2005001966 W 20051219; AR P050105335 A 20051219; EP 05819128 A 20051219; JP 2007548144 A 20051219; TW 94145647 A 20051221; US 72176705 A 20051219