Global Patent Index - EP 1838662 A1

EP 1838662 A1 2007-10-03 - SQUARIC ACID DERIVATIVES

Title (en)

SQUARIC ACID DERIVATIVES

Title (de)

QUADRATSÄUREDERIVATE

Title (fr)

DERIVES D'ACIDE QUADRATIQUE

Publication

EP 1838662 A1 (DE)

Application

EP 05849991 A

Priority

  • EP 2005013225 W
  • DE 102005001053 A

Abstract (en)

[origin: WO2006072354A1] The invention relates to novel squaric acid compounds of formula (I) wherein R, R<SUP>l</SUP>, R<SUP>1'</SUP>, R<SUP>2</SUP> and X have the designations cited in patent claim (1). Said compounds are SGK inhibitors and can be used to treat SGK-related diseases and illnesses such as diabetes, obesity, metabolic syndrome (dyslipidaemia), systemic and pulmonal hypertonia, cardiovascular diseases and kidney diseases, and generally all types of fibroses and inflammatory processes.

IPC 8 full level (invention and additional information)

C07C 225/20 (2006.01); A61K 31/135 (2006.01); A61P 3/00 (2006.01); A61P 9/00 (2006.01); A61P 13/12 (2006.01)

CPC (invention and additional information)

C07C 225/20 (2013.01); C07C 225/22 (2013.01); C07C 255/59 (2013.01); C07C 311/37 (2013.01); C07C 311/39 (2013.01); C07C 2601/02 (2017.05); C07C 2601/04 (2017.05)

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

EPO simple patent family

WO 2006072354 A1 20060713; AR 056636 A1 20071017; AU 2005324119 A1 20060713; CA 2594388 A1 20060713; DE 102005001053 A1 20060720; EP 1838662 A1 20071003; JP 2008526790 A 20080724; US 2008262096 A1 20081023

INPADOC legal status


2010-10-27 [18D] DEEMED TO BE WITHDRAWN

- Effective date: 20100429

2010-01-20 [17Q] FIRST EXAMINATION REPORT

- Effective date: 20091218

2008-04-16 [DAX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT (TO ANY COUNTRY) DELETED

2007-10-03 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20070509

2007-10-03 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR