EP 1846381 A2 20071024 - HETEROARYLACETAMIDES AS FACTOR Xa INHIBITORS
Title (en)
HETEROARYLACETAMIDES AS FACTOR Xa INHIBITORS
Title (de)
HETEROARYLACETAMIDE ALS FAKTOR Xa INHIBITOREN
Title (fr)
HETEROARYLACETAMIDES COMME INHIBITEURS DU FACTEUR Xa
Publication
Application
Priority
- EP 2005013460 W 20051214
- EP 04106943 A 20041223
- EP 05817940 A 20051214
Abstract (en)
[origin: WO2006066778A2] The invention is concerned with novel heteroarylacetamides of formula (I) R<SUP>d</SUP>-C(O)-N(R<SUP>e</SUP>)-R<SUP>c</SUP>-CH<SUB>2</SUB>-C(O)-N(R<SUP>a</SUP>)(R<SUP>b</SUP>), wherein R<SUP>a</SUP> to R<SUP>e</SUP> are as defined in the description and in the claims, as well as physiologically acceptable salts thereof. These compounds inhibit the coagulation factor Xa and can be used as medicaments.
IPC 8 full level
C07D 277/46 (2006.01); C07D 401/10 (2006.01); C07D 409/06 (2006.01); C07D 409/14 (2006.01); C07D 417/06 (2006.01); C07D 417/10 (2006.01); C07D 417/14 (2006.01)
CPC (source: EP KR US)
A61P 7/02 (2018.01 - EP); A61P 9/00 (2018.01 - EP); A61P 9/04 (2018.01 - EP); A61P 9/10 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 35/00 (2018.01 - EP); C07D 277/46 (2013.01 - EP US); C07D 401/10 (2013.01 - EP US); C07D 409/06 (2013.01 - EP KR US); C07D 409/14 (2013.01 - EP US); C07D 417/06 (2013.01 - EP KR US); C07D 417/10 (2013.01 - EP KR US); C07D 417/14 (2013.01 - EP KR US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2006066778 A2 20060629; WO 2006066778 A3 20060810; AT E396979 T1 20080615; AU 2005318538 A1 20060629; BR PI0519439 A2 20090120; CA 2591117 A1 20060629; CA 2591117 C 20140422; CN 101124208 A 20080213; CN 101124208 B 20110706; DE 602005007270 D1 20080710; EP 1846381 A2 20071024; EP 1846381 B1 20080528; ES 2308581 T3 20081201; JP 2008525337 A 20080717; JP 4954895 B2 20120620; KR 20070089245 A 20070830; MX 2007007486 A 20070720; RU 2007128065 A 20090127; US 2006142362 A1 20060629; US 2008146550 A1 20080619; US 7361672 B2 20080422; US 7718659 B2 20100518
DOCDB simple family (application)
EP 2005013460 W 20051214; AT 05817940 T 20051214; AU 2005318538 A 20051214; BR PI0519439 A 20051214; CA 2591117 A 20051214; CN 200580048547 A 20051214; DE 602005007270 T 20051214; EP 05817940 A 20051214; ES 05817940 T 20051214; JP 2007547282 A 20051214; KR 20077016782 A 20070720; MX 2007007486 A 20051214; RU 2007128065 A 20051214; US 2512408 A 20080204; US 30156005 A 20051213